SCHEMBL9702109

SCHEMBL9702109

COc1ccc2cc(C(N)=O)ccc2c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.70
PARP10 Q53GL7 3/20 0.68
PARP1 P09874 2/20 0.68
PARP4 Q9UKK3 2/20 0.68
CA1 P00915 1/20 0.68
CA2 P00918 1/20 0.68
PARP2 Q9UGN5 1/20 0.68
HPGDS O60760 1/20 0.64
PLAU P00749 4/20 0.62
CYP11B1 P15538 1/20 0.59
CYP11B2 P19099 1/20 0.59
ALDH1A1 P00352 2/20 0.58
CYP1A2 P05177 2/20 0.58
HPGD P15428 1/20 0.58
CYP2C19 P33261 1/20 0.58
HSD17B10 Q99714 1/20 0.58
LCK P06239 1/20 0.58
PLAT P00750 2/20 0.55
PLG P00747 1/20 0.55
MAP4K4 O95819 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11810869 0.84 KDM4E (0.75) KDM4ECA1CA2PLAUALDH1A1
SCHEMBL2363489 0.83 LCK (0.78) KDM4EPARP10PARP1PARP4CA1
SCHEMBL7567274 0.83 LCK (0.61) KDM4EPARP10PARP1PARP4CA1
SCHEMBL29793856 0.82 KDM4E (0.72) KDM4EPLAUCYP11B1CYP11B2ALDH1A1
SCHEMBL34463427 0.82 KDM4E (1.00) KDM4ECA1CA2PLAUALDH1A1
SCHEMBL246511 0.82 KDM4E (0.72) KDM4EPLAUCYP11B1CYP11B2ALDH1A1
SCHEMBL8132 0.82 KDM4E (1.00) KDM4ECA1CA2PLAUALDH1A1
SCHEMBL3659867 0.82 CYP11B1 (0.68) PARP1HPGDSPLAUCYP11B1CYP11B2
SCHEMBL3922405 0.81 LCK (0.55) KDM4EPARP10PARP1PARP4CA1
SCHEMBL201761 0.81 PARP10 (1.00) PARP10PARP1PARP4CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010108651-A1 SUBSTITUTED SPIRO-AMIDE COMPOUNDS Grünenthal GmbH (DE) 2010-09-30 WO disclosed
EP-0221677-B1 P-AMINOPHENOLS, DERIVATIVES THEREOF AND USE FOR MANUFACTURE OF A MEDICAMENT E.R. Squibb & Sons, Inc. (US) 1992-09-09 EP disclosed
US-4910208-A Skin disorders, antiinflammatory agent E. R. SQUIBB & SONS, INC. (US) 1990-03-20 US disclosed
US-4814454-A ANTIALLERGENS, ANTIINFLAMMATORY E. R. SQUIBB & SONS, INC. (US) 1989-03-21 US disclosed
EP-0221677-A2 p-Aminophenols, derivatives thereof and use for manufacture of a medicament E.R. Squibb & Sons, Inc. (US) 1987-05-13 EP disclosed