SCHEMBL9702533

SCHEMBL9702533

O=C(O)Cn1ccc2cc(Cl)ccc21

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.60
KMO O15229 3/20 0.55
OXER1 Q8TDS5 2/20 0.55
HTR2A P28223 1/20 0.53
HTR2C P28335 1/20 0.53
RHEB Q15382 1/20 0.52
KRAS P01116 2/20 0.51
ACLY P53396 2/20 0.49
PTGDR2 Q9Y5Y4 1/20 0.48
PPARD Q03181 3/20 0.47
PPARG P37231 2/20 0.47
PPARA Q07869 2/20 0.47
NPY5R Q15761 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29957878 0.87 KMO (0.72) KMT2AKMOOXER1RHEBACLY
SCHEMBL1576364 0.87 KMO (0.72) KMT2AKMOOXER1RHEBACLY
SCHEMBL2006946 0.85 HTR2A (0.55) KMT2AKMOOXER1HTR2AHTR2C
SCHEMBL9701399 0.85 HTR2A (0.55) KMT2AKMOOXER1HTR2AHTR2C
SCHEMBL1576323 0.84 KMO (0.78) KMOOXER1HTR2AHTR2CACLY
SCHEMBL416786 0.81 KMO (0.65) KMOOXER1HTR2AHTR2CACLY
SCHEMBL27591506 0.81 HTR2A (0.58) KMOOXER1HTR2AHTR2CKRAS
SCHEMBL4234811 0.81 KMT2A (0.62) KMT2APPARDPPARGPPARA
SCHEMBL30103437 0.81 KMT2A (0.62) KMT2APPARDPPARGPPARA
SCHEMBL29174329 0.80 KMO (0.63) KMT2AKMOOXER1RHEBACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018065607-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2018-04-12 WO disclosed
EP-3305781-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN-RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum (DE) 2018-04-11 EP disclosed
EP-3305781-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN-RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum (DE) 2018-04-11 EP disclosed
US-5132319-A Antiasthmatic, antiinflammatory, antiallergen and cytoprotective agents MERCK FROSST CANADA, INC. (CA) 1992-07-21 US disclosed