SCHEMBL9702567

SCHEMBL9702567

CC(NC(=O)O)C(=O)NC(CNCC=CC(=O)OCCc1c[nH]c2ccccc12)Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NMBR P28336 6/20 0.47
KMT2A Q03164 2/20 0.47
ALDH1A1 P00352 2/20 0.47
CYP3A4 P08684 2/20 0.47
MAPT P10636 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47
MAPK1 P28482 1/20 0.47
HSD17B10 Q99714 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
CTSL P07711 1/20 0.44
ACE P12821 1/20 0.41
TP53 P04637 1/20 0.41
MDM2 Q00987 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9702562 0.85 NMBR (0.47) NMBRALDH1A1CYP3A4MAPTCTSL
SCHEMBL9540282 0.75 TACR1 (0.50)
SCHEMBL9540278 0.75 TACR1 (0.50)
SCHEMBL23100729 0.69 ECE1 (0.65) KMT2AALDH1A1CYP3A4MAPTKDM4E
SCHEMBL23100728 0.69 ECE1 (0.65) KMT2AALDH1A1CYP3A4MAPTKDM4E
SCHEMBL8895674 0.67 CTSL (0.55) KMT2AALDH1A1CYP3A4MAPTKDM4E
SCHEMBL8098291 0.67 NMBR (0.69) NMBRMAPTACE
SCHEMBL12052755 0.67 NMBR (0.69) NMBRMAPTACE
SCHEMBL12062839 0.67 NMBR (0.69) NMBRMAPTACE
SCHEMBL5380211 0.67 NMBR (0.69) NMBRMAPTACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992004038-A1 PRO-DRUGS FOR CCK ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1992-03-19 WO disclosed