SCHEMBL9703681

SCHEMBL9703681

Cc1cccc2c1C(c1ccccc1)=NN(c1ccc(F)cc1)C(=O)N2C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 3/20 0.38
BACE1 P56817 2/20 0.36
APP P05067 1/20 0.35
GABRA1 P14867 2/20 0.35
GABRG2 P18507 2/20 0.35
GABRB3 P28472 2/20 0.35
GABRA5 P31644 2/20 0.35
GABRA3 P34903 2/20 0.35
GABRA2 P47869 2/20 0.35
GABRB2 P47870 2/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRA4 P48169 1/20 0.35
GABRE P78334 1/20 0.35
GABRA6 Q16445 1/20 0.35
GABRG1 Q8N1C3 1/20 0.35
GABRG3 Q99928 1/20 0.35
GABRQ Q9UN88 1/20 0.35
CES2 O00748 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9705387 0.88 CCKBR (0.38) CCKBRBACE1APPGABRA1GABRG2
SCHEMBL9703566 0.83 CCKBR (0.38) CCKBRGABRA1GABRG2GABRB3GABRA5
SCHEMBL9703671 0.66 PTH1R (0.49) CCKBRGABRA1GABRG2GABRB3GABRA5
Dimethylamine SCHEMBL9651824 0.65 MAPT (0.40) CCKBRAPPCES2KDM4ENPC1
SCHEMBL9651820 0.64 KMT2A (0.71) KDM4ENPC1ALDH1A1MAPTRAB9A
SCHEMBL9651814 0.64 KMT2A (0.71) KDM4ENPC1ALDH1A1MAPTRAB9A
SCHEMBL9702894 0.63 CCKBR (0.49) CCKBRGABRA1GABRG2GABRB3GABRA5
SCHEMBL9653091 0.62 MEN1 (0.58) KDM4ENPC1ALDH1A1MAPTRAB9A
SCHEMBL6730982 0.61 APP (0.46) APPCES2PTGS1KDM4ENPC1
SCHEMBL8555730 0.59 MAOB (0.39) SLC6A4KDM4ENPC1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091381-A Detection of peripheral benzodiazepine receptor activity in cell or tissue by labelled compounds using radioisotopes or cytoxic agents BIOMEASURE, INC. (US) 1992-02-25 US disclosed