SCHEMBL9703840

SCHEMBL9703840

c1cc(N2CCOCC2)c2cc[nH]c2c1

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.69
HTR6 P50406 1/20 0.69
DRD2 P14416 1/20 0.57
DRD4 P21917 1/20 0.57
DRD3 P35462 1/20 0.57
GAA P10253 6/20 0.53
MAPT P10636 3/20 0.52
GOT1 P17174 8/20 0.51
RECQL P46063 1/20 0.51
PIK3CD O00329 1/20 0.51
HTR1A P08908 1/20 0.49
PIK3CA P42336 1/20 0.47
MTOR P42345 1/20 0.47
ATR Q13535 1/20 0.46
MEN1 O00255 1/20 0.46
GFER P55789 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29941044 1.00 ADRB1 (0.69) ADRB1HTR6DRD2DRD4DRD3
SCHEMBL20581870 0.84 ADRB1 (0.75) ADRB1HTR6DRD2DRD4DRD3
SCHEMBL30160211 0.83 ADRB1 (0.73) ADRB1HTR6DRD2DRD4DRD3
SCHEMBL8861994 0.83 ADRB1 (0.73) ADRB1HTR6DRD2DRD4DRD3
SCHEMBL1012802 0.81 ADRB1 (1.00) ADRB1HTR6DRD2DRD4DRD3
Hydrochloric Acid SCHEMBL6730585 0.80 ADRB1 (0.97) ADRB1HTR6DRD2DRD4DRD3
Hydrochloric Acid SCHEMBL4662618 0.80 ADRB1 (0.97) ADRB1HTR6DRD2DRD4DRD3
SCHEMBL4306478 0.80 ADRB1 (0.69) ADRB1HTR6DRD2DRD4DRD3
SCHEMBL5430904 0.80 ADRB1 (0.69) ADRB1HTR6DRD2DRD4DRD3
SCHEMBL9260887 0.80 ADRB1 (0.46) ADRB1HTR6DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0230179-B1 4-MORPHOLINYL 1H-INDOLE DERIVATIVES, THEIR SALTS, PROCESS AND INTERMEDIATES OF PREPARATION, USE AS THERAPEUTIC AGENTS, COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1992-09-30 EP claimed
US-4699907-A ANTIISCHEMIC, HYPOTENSIVE AGENTS ROUSSEL UCLAF (FR) 1987-10-13 US claimed
US-20250263760-A1 MODIFIED BACTERIA FOR PRODUCTION OF NITROAROMATICS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2025-08-21 US disclosed
US-12319946-B2 Methods for producing modified bacteria for production of nitroaromatics UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2025-06-03 US disclosed
US-20240229090-A1 MODIFIED BACTERIA FOR PRODUCTION OF NITROAROMATICS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2024-07-11 US disclosed
US-20240229090-A1 MODIFIED BACTERIA FOR PRODUCTION OF NITROAROMATICS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2024-07-11 US disclosed
US-20240229090-A1 MODIFIED BACTERIA FOR PRODUCTION OF NITROAROMATICS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2024-07-11 US disclosed
US-11879144-B2 Modified bacteria for production of nitroaromatics UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2024-01-23 US disclosed
US-20230287466-A1 MODIFIED BACTERIA FOR PRODUCTION OF NITROAROMATICS UNIVERSITY OF FLORIDA RESEARCH (US) 2023-09-14 US disclosed
US-20230287466-A1 MODIFIED BACTERIA FOR PRODUCTION OF NITROAROMATICS UNIVERSITY OF FLORIDA RESEARCH (US) 2023-09-14 US disclosed
US-20230287466-A1 MODIFIED BACTERIA FOR PRODUCTION OF NITROAROMATICS UNIVERSITY OF FLORIDA RESEARCH (US) 2023-09-14 US disclosed
WO-2016134145-A9 ARTIFICIAL SELF-SUFFICIENT CYTOCHROME P450S UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2017-02-16 WO disclosed
WO-2016134145-A9 ARTIFICIAL SELF-SUFFICIENT CYTOCHROME P450S UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2017-02-16 WO disclosed
WO-2016134145-A2 ARTIFICIAL SELF-SUFFICIENT CYTOCHROME P450S UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2016-08-25 WO disclosed
WO-2016134145-A2 ARTIFICIAL SELF-SUFFICIENT CYTOCHROME P450S UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2016-08-25 WO disclosed
US-4736042-A CHEMICAL INTERMEDIATES ROUSSEL UCLAF (FR) 1988-04-05 US disclosed
US-4736042-A CHEMICAL INTERMEDIATES ROUSSEL UCLAF (FR) 1988-04-05 US disclosed
US-4699907-A ANTIISCHEMIC, HYPOTENSIVE AGENTS ROUSSEL UCLAF (FR) 1987-10-13 US disclosed
US-4699907-A ANTIISCHEMIC, HYPOTENSIVE AGENTS ROUSSEL UCLAF (FR) 1987-10-13 US disclosed
US-4699907-A ANTIISCHEMIC, HYPOTENSIVE AGENTS ROUSSEL UCLAF (FR) 1987-10-13 US disclosed