SCHEMBL970522

SCHEMBL970522

O=CNc1c[nH]c2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 2/20 0.53
CYP2A6 P11509 1/20 0.53
STING1 Q86WV6 9/20 0.45
GPR84 Q9NQS5 2/20 0.44
IMPDH1 P20839 1/20 0.44
ATM Q13315 1/20 0.44
PABPC1 P11940 1/20 0.43
MEN1 O00255 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAPT P10636 1/20 0.42
AHR P35869 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27963053 0.87 IMPDH2 (0.49) IMPDH2CYP2A6STING1GPR84IMPDH1
SCHEMBL28156918 0.81 CYP2A6 (0.50) IMPDH2CYP2A6STING1GPR84ATM
SCHEMBL28743536 0.81 IMPDH2 (0.44) IMPDH2CYP2A6STING1GPR84IMPDH1
SCHEMBL2855201 0.81 MEN1 (0.47) IMPDH2CYP2A6STING1GPR84IMPDH1
SCHEMBL28346693 0.78 STING1 (0.49) IMPDH2CYP2A6STING1GPR84ATM
SCHEMBL6654114 0.77 ATM (0.52) IMPDH2CYP2A6STING1GPR84IMPDH1
SCHEMBL22299626 0.77 CYP2A6 (0.49) IMPDH2CYP2A6STING1GPR84MEN1
SCHEMBL349436 0.76 MAPK1 (0.51) PABPC1AHR
SCHEMBL747027 0.75 STING1 (0.55) IMPDH2CYP2A6STING1GPR84
SCHEMBL27629215 0.75 NPC1 (0.48) IMPDH2CYP2A6STING1GPR84IMPDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 196 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119306650-A Preparation method of indole carboxamide compound 西安睿舒维生物医药科技有限公司 2025-01-14 CN claimed
CN-115260080-A Preparation method of indole-3-carboxamide compound 浙江理工大学 2022-11-01 CN claimed
CN-109824574-B Indole-3-carboxamides and their use 沈阳药科大学 2021-12-28 CN claimed
CN-108101828-B 3-indolyl formamide compound and preparation method thereof 西华师范大学 2021-05-04 CN claimed
CN-110475557-A (R)-N- ((4- methoxyl group-6- methyl-2- oxo-1,2- dihydropyridine-3- base) methyl)-2- methyl-1-(1- (1- (2,2,2- trifluoroethyl) piperidin-4-yl) ethyl) and-1H- indoles-3- formamide solid dispersions CONSTELLATION PHARMACEUTICALS INC 2019-11-19 CN claimed
CN-110022869-A For skin and/or the serotonin 1B receptor stimulators of hair reparation 巴斯德研究院 2019-07-16 CN claimed
CN-106478662-B 5-HT3 receptor antagonist 武田药品工业株式会社 2019-07-02 CN claimed
CN-109824574-A Indoles -3- Carbox amide and its application 沈阳药科大学 2019-05-31 CN claimed
CN-106946761-B Indole carboxamides class compound and its application 沈阳药科大学 2019-05-03 CN claimed
CN-106459030-B Replace tropane derivatives 东亚荣养株式会社 2019-01-29 CN claimed
CN-108348486-A 5-hydroxytryptamine 1B receptor agonists as promoters for satellite cell self-renewal and/or differentiation 巴斯德研究院 2018-07-31 CN claimed
CN-108329253-A Preceding neurogenic compounds 得克萨斯州大学系统董事会 2018-07-27 CN claimed
CN-105198789-B Substitute 3- indoles Bcl-2 protein inhibitors and preparation method and application 山东大学 2018-06-05 CN claimed
CN-108026073-A Fluoroindole derivatives as muscarinic M 1 receptor forward direction allosteric modulators 苏文生命科学有限公司 2018-05-11 CN claimed
CN-105612150-B Sulfonylindole derivatives and process for producing the same 株式会社大熊制药 2018-04-10 CN claimed
CN-105073741-B Phthalazinones and isoquinolinones as ROCK inhibitors 百时美施贵宝公司 2017-08-08 CN claimed
CN-106946761-A Indole carboxamides class compound and its application 沈阳药科大学 2017-07-14 CN claimed
CN-104744460-B β carbolines, dihydro β carbolines and tetrahydro-beta-carboline alcaloid-derivatives and preparation method thereof and the application in terms of preventing and treating plant virus, sterilization, desinsection 南开大学 2017-06-16 CN claimed
CN-119306650-A Preparation method of indole carboxamide compound 西安睿舒维生物医药科技有限公司 2025-01-14 CN disclosed
US-5212195-A Substituted indole antagonists derivatives which are angiotensin II SYNTEX (U.S.A.) INC. (US) 1993-05-18 US disclosed