SCHEMBL9705299

SCHEMBL9705299

O=C(Nc1nc2c(ncn2[C@@H]2O[C@H](COC(c3ccccc3)(c3ccccc3)c3ccccc3)[C@@H](O)[C@H]2OC(c2ccccc2)(c2ccccc2)c2ccccc2)c(=O)[nH]1)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TYMP P19971 14/20 0.56
TAS1R3 Q7RTX0 2/20 0.52
TAS1R1 Q7RTX1 2/20 0.52
NT5E P21589 2/20 0.47
HINT1 P49773 1/20 0.46
IMPDH2 P12268 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9706215 0.92 TAS1R3 (0.60) TYMPTAS1R3TAS1R1NT5EHINT1
SCHEMBL9705378 0.90 TYMP (0.54) TYMPTAS1R3TAS1R1NT5EHINT1
SCHEMBL9705652 0.89 TYMP (0.58) TYMPTAS1R3TAS1R1NT5EHINT1
SCHEMBL30689445 0.88 TYMP (0.70) TYMPTAS1R3TAS1R1HINT1IMPDH2
SCHEMBL34234 0.85 TYMP (0.64) TYMPTAS1R3TAS1R1NT5EHINT1
SCHEMBL8613074 0.85 TYMP (0.49) TYMPNT5E
SCHEMBL9705754 0.84 TYMP (0.54) TYMPTAS1R3TAS1R1NT5EHINT1
SCHEMBL9705666 0.83 TYMP (0.58) TYMP
SCHEMBL6514428 0.82 TYMP (0.57) TYMPTAS1R3TAS1R1NT5EHINT1
SCHEMBL30689462 0.82 TYMP (0.53) TYMPTAS1R3TAS1R1NT5EHINT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992011276-A1 NOVEL SYNTHESIS OF 2'-'UP' FLUORINATED 2''-DEOXY-ARABINOFURANOSYLPURINES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-07-09 WO claimed
WO-1992011276-A1 NOVEL SYNTHESIS OF 2'-'UP' FLUORINATED 2''-DEOXY-ARABINOFURANOSYLPURINES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-07-09 WO disclosed