SCHEMBL9705784

SCHEMBL9705784

CCCCc1nc(=O)c2ccncc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.51
GSK3B P49841 1/20 0.49
PARP1 P09874 2/20 0.46
KDM5A P29375 4/20 0.45
TRPV1 Q8NER1 3/20 0.44
ADORA3 P0DMS8 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
KDM5B Q9UGL1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27126276 0.85 KDM5A (0.52) KDM4CPARP1KDM5AADORA3ADORA2A
SCHEMBL8501957 0.81 PARP1 (0.60) PARP1
SCHEMBL9853656 0.79 KDM4C (0.49) KDM4CGSK3BPARP1
Alcohol SCHEMBL27310243 0.77 PARP1 (0.56) PARP1
SCHEMBL9376294 0.77 KMT2A (0.54) GSK3BPARP1
SCHEMBL1586540 0.77 PARP1 (0.55) PARP1
SCHEMBL8566027 0.76 KDM4C (0.52) KDM4CGSK3BPARP1
SCHEMBL9706231 0.75 PARP1 (0.54) GSK3BPARP1
SCHEMBL9052175 0.74 MAPT (0.59) GSK3BPARP1
SCHEMBL31338639 0.73 PARP1 (0.49) KDM4CGSK3BPARP1KDM5AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481614-A1 Substituted pyridopyrimidinones and related heterocycles as angiotensin II antagonists MERCK & CO. INC. (US) 1992-04-22 EP disclosed