SCHEMBL9705864

SCHEMBL9705864

CC(=O)N1c2ncccc2NC(=O)c2cccnc21

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.58
CHRM2 P08172 4/20 0.53
LMNA P02545 2/20 0.53
CHRM1 P11229 2/20 0.53
USP2 O75604 1/20 0.53
ALDH1A1 P00352 1/20 0.53
CYP1A2 P05177 1/20 0.53
CHRM4 P08173 1/20 0.53
CHRM5 P08912 1/20 0.53
CYP2D6 P10635 1/20 0.53
CHRM3 P20309 1/20 0.53
GMNN O75496 1/20 0.52
APEX1 P27695 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4541695 0.88 RAB9A (0.72) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL9596507 0.77 RAB9A (0.61) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL9596882 0.77 RAB9A (0.76) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL26060354 0.77 RAB9A (0.67) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL11196254 0.77 RAB9A (0.67) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL10392149 0.76 RAB9A (0.70) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL8304745 0.75 CYP1A2 (0.49) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL8300334 0.75 RAB9A (0.50) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL7553424 0.75 RAB9A (0.80) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL10968958 0.75 RAB9A (0.68) RAB9ACHRM2LMNACHRM1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0482481-A1 Method for the preparation of 5,11-dihydro-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepines BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 1992-04-29 EP disclosed