SCHEMBL9705868

SCHEMBL9705868

CCN1c2ncccc2NC(=O)c2cc(C)cnc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.45
CYP2C19 P33261 3/20 0.45
CYP3A4 P08684 2/20 0.45
CYP1A2 P05177 3/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 2/20 0.41
NPC1 O15118 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
MCL1 Q07820 1/20 0.41
CHRM2 P08172 3/20 0.40
ROS1 P08922 1/20 0.39
CDK5 Q00535 1/20 0.39
ACVR1 Q04771 1/20 0.39
LRRK2 Q5S007 1/20 0.39
USP2 O75604 1/20 0.39
LMNA P02545 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM5 P08912 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9704218 0.90 CYP2C9 (0.47) CYP2C9CYP2C19CYP3A4CYP1A2RAB9A
SCHEMBL4031265 0.87 RAB9A (0.43) CYP2C9CYP2C19CYP3A4CYP1A2RAB9A
SCHEMBL8300334 0.86 RAB9A (0.50) CYP1A2RAB9ASMN1; SMN2ALDH1A1CHRM2
SCHEMBL6959718 0.83 MEN1 (0.43) CYP2C9CYP2C19CYP3A4RAB9AALDH1A1
SCHEMBL14418888 0.83 CYP3A4 (0.46) CYP2C9CYP2C19CYP3A4CYP1A2RAB9A
SCHEMBL6963218 0.83 CYP3A4 (0.46) CYP2C9CYP2C19CYP3A4CYP1A2RAB9A
SCHEMBL14425195 0.82 CYP3A4 (0.45) CYP2C9CYP2C19CYP3A4CYP1A2RAB9A
SCHEMBL9703875 0.82 CYP2C9 (0.42) CYP2C9CYP2C19CYP3A4CYP1A2RAB9A
SCHEMBL14418887 0.81 CYP3A4 (0.48) CYP2C9CYP2C19CYP3A4CYP1A2RAB9A
SCHEMBL9704536 0.79 RAB9A (0.42) CYP2C9CYP2C19CYP3A4CYP1A2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0482481-A1 Method for the preparation of 5,11-dihydro-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepines BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 1992-04-29 EP disclosed