SCHEMBL9707639

SCHEMBL9707639

COCCn1c(=O)n(CC(=O)OC)c(=O)c2c1nc(CC(C)(C)C)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 6/20 0.40
AGTR2 P50052 3/20 0.40
KMT2A Q03164 2/20 0.39
HTT P42858 1/20 0.38
ALDH1A1 P00352 2/20 0.38
POLB P06746 1/20 0.37
MEN1 O00255 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
PPARG P37231 1/20 0.36
TP53 P04637 1/20 0.36
TSHR P16473 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708964 0.98 AGTR1 (0.40) AGTR1AGTR2KMT2AHTTALDH1A1
SCHEMBL9707900 0.95 AGTR1 (0.43) AGTR1AGTR2KMT2AMEN1CYP2C9
SCHEMBL9708108 0.94 AGTR1 (0.44) AGTR1AGTR2KMT2AMEN1CYP2C9
SCHEMBL9708498 0.92 AGTR1 (0.43) AGTR1AGTR2KMT2AALDH1A1MEN1
SCHEMBL9707449 0.92 KMT2A (0.45) AGTR1AGTR2KMT2AHTTALDH1A1
SCHEMBL9707642 0.92 AGTR1 (0.43) AGTR1AGTR2KMT2APPARGADORA3
SCHEMBL9707542 0.91 AGTR1 (0.43) AGTR1AGTR2KMT2APPARG
SCHEMBL9708531 0.91 AGTR1 (0.40) AGTR1AGTR2KMT2AMEN1CYP2C9
SCHEMBL9708107 0.91 AGTR1 (0.47) AGTR1AGTR2KMT2APPARG
SCHEMBL9708139 0.91 TSHR (0.42) AGTR1AGTR2KMT2AHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed