SCHEMBL9707774

SCHEMBL9707774

COC(C)n1c(=O)[nH]c(=O)c2c1nc(C1CCCCC1)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.46
AGTR1 P30556 5/20 0.40
AGTR2 P50052 3/20 0.40
NPSR1 Q6W5P4 3/20 0.38
POLB P06746 2/20 0.38
MAPK1 P28482 1/20 0.38
BLM P54132 1/20 0.38
CTDSP1 Q9GZU7 1/20 0.38
MEN1 O00255 3/20 0.37
RAB9A P51151 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
PPARG P37231 4/20 0.35
PDE5A O76074 1/20 0.34
PDE1A P54750 1/20 0.34
PDE1B Q01064 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708539 0.90 AGTR1 (0.40) KMT2AAGTR1AGTR2NPSR1POLB
SCHEMBL9708436 0.90 KMT2A (0.48) KMT2AAGTR1AGTR2NPSR1POLB
SCHEMBL9708507 0.89 AGTR1 (0.39) KMT2AAGTR1AGTR2NPSR1POLB
SCHEMBL9708478 0.88 PDE5A (0.39) KMT2AAGTR1AGTR2NPSR1POLB
SCHEMBL9708405 0.88 AGTR1 (0.39) KMT2AAGTR1AGTR2NPSR1POLB
SCHEMBL9707885 0.87 KMT2A (0.52) KMT2AAGTR1AGTR2NPSR1POLB
SCHEMBL9708383 0.87 PDE5A (0.39) KMT2AAGTR1AGTR2NPSR1POLB
SCHEMBL9708565 0.87 KMT2A (0.55) KMT2AAGTR1AGTR2NPSR1POLB
SCHEMBL9708060 0.87 MAPK1 (0.41) KMT2AAGTR1AGTR2NPSR1POLB
SCHEMBL9707827 0.86 AGTR1 (0.38) KMT2AAGTR1AGTR2NPSR1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed