SCHEMBL9708792

SCHEMBL9708792

COC(=O)Cn1c(=O)[nH]c(=O)c2c1nc(C1CCCCC1)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.50
MEN1 O00255 4/20 0.41
POLB P06746 1/20 0.41
RAB9A P51151 1/20 0.41
AGTR1 P30556 5/20 0.40
AGTR2 P50052 4/20 0.40
PPARG P37231 3/20 0.40
NPSR1 Q6W5P4 2/20 0.40
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
TPH1 P17752 1/20 0.39
TPH2 Q8IWU9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707400 0.90 AGTR1 (0.42) KMT2APOLBAGTR1AGTR2PPARG
SCHEMBL9707883 0.90 PPARG (0.42) KMT2AAGTR1AGTR2PPARG
SCHEMBL9708284 0.90 KMT2A (0.54) KMT2AMEN1POLBRAB9AAGTR1
SCHEMBL9707780 0.89 KMT2A (0.53) KMT2AMEN1POLBRAB9AAGTR1
SCHEMBL9707644 0.89 KMT2A (0.41) KMT2AMEN1POLBAGTR1AGTR2
SCHEMBL9708457 0.88 KMT2A (0.55) KMT2AMEN1POLBRAB9AAGTR1
SCHEMBL9708763 0.88 PDE5A (0.43) KMT2AAGTR1AGTR2PPARG
SCHEMBL9707886 0.88 PDE5A (0.43) KMT2AAGTR1AGTR2PPARG
SCHEMBL9708854 0.88 KMT2A (0.41) KMT2APOLBAGTR1AGTR2PPARG
SCHEMBL9707885 0.87 KMT2A (0.52) KMT2AMEN1POLBRAB9AAGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed