SCHEMBL9708961

SCHEMBL9708961

COC(=O)Cn1c(=O)n(C(C)OC)c(=O)c2c1nc(CC(C)(C)C)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 6/20 0.40
AGTR2 P50052 6/20 0.40
PPARG P37231 3/20 0.37
TP53 P04637 1/20 0.34
TSHR P16473 1/20 0.34
AVPR2 P30518 1/20 0.34
AVPR1A P37288 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707631 0.95 AGTR1 (0.40) AGTR1AGTR2PPARGTP53TSHR
SCHEMBL9708688 0.93 AGTR1 (0.39) AGTR1AGTR2PPARG
SCHEMBL9707805 0.92 AGTR1 (0.43) AGTR1AGTR2PPARGKMT2A
SCHEMBL9707900 0.91 AGTR1 (0.43) AGTR1AGTR2PPARGTP53TSHR
SCHEMBL9707676 0.91 AGTR1 (0.46) AGTR1AGTR2PPARG
SCHEMBL9708255 0.91 AGTR1 (0.35) AGTR1AGTR2
SCHEMBL9707537 0.91 AGTR1 (0.36) AGTR1AGTR2PPARG
SCHEMBL9708632 0.90 AGTR1 (0.40) AGTR1AGTR2PPARGKMT2A
SCHEMBL9708139 0.90 TSHR (0.42) AGTR1AGTR2PPARGTP53TSHR
SCHEMBL9707436 0.90 AGTR1 (0.52) AGTR1AGTR2PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed