SCHEMBL9709031

SCHEMBL9709031

Nc1ccc2c(c1N)NC(=O)CC2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 1/20 0.50
NPC1 O15118 1/20 0.42
MAPK13 O15264 1/20 0.42
MAPK12 P53778 1/20 0.42
MAPK11 Q15759 1/20 0.42
MAPK14 Q16539 1/20 0.42
SRD5A1 P18405 5/20 0.40
CRBN Q96SW2 3/20 0.39
CYP11B1 P15538 4/20 0.35
CYP11B2 P19099 4/20 0.35
CYP19A1 P11511 3/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
POLB P06746 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KDM4E B2RXH2 2/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3593739 0.78 NPC1 (0.50) CA9NPC1MAPK13MAPK12MAPK11
SCHEMBL27140279 0.72 CA9 (0.42) CA9NPC1MAPK13MAPK12MAPK11
SCHEMBL27148030 0.71 NPC1 (0.41) CA9NPC1MAPK13MAPK12MAPK11
SCHEMBL30062471 0.71 SRD5A1 (0.41) CA9NPC1MAPK13MAPK12MAPK11
SCHEMBL852124 0.71 PARP1 (0.47) CA9NPC1MAPK13MAPK12MAPK11
SCHEMBL30893045 0.71 NPC1 (0.41) CA9NPC1MAPK13MAPK12MAPK11
SCHEMBL27139794 0.71 SRD5A1 (0.41) CA9NPC1MAPK13MAPK12MAPK11
SCHEMBL21468468 0.70 MAPT (0.39) CA9NPC1CRBNALDH1A1MAPT
SCHEMBL9379056 0.69 CYP19A1 (0.39) CYP19A1ALDH1A1KDM4ELMNAHPGD
SCHEMBL18513655 0.68 CA9 (0.42) CA9NPC1MAPK13MAPK12MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0473963-A1 Pyrrolobenzimidazoles, imidazobenzoxazinones, and imidazoquinolones, processes for their preparation and their use as well as compositions containing these compounds Beiersdorf-Lilly GmbH (DE) 1992-03-11 EP disclosed