SCHEMBL9709721

SCHEMBL9709721

CCCc1cc(NC(=O)OC(C)(C)C)c2ccccc2n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.54
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
HTT P42858 2/20 0.50
GAA P10253 3/20 0.49
RAB9A P51151 2/20 0.49
NPC1 O15118 1/20 0.49
SREBF2 Q12772 1/20 0.47
ALDH1A1 P00352 3/20 0.47
HPGD P15428 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
TOP2A P11388 1/20 0.46
TOP2B Q02880 1/20 0.46
TLR7 Q9NYK1 1/20 0.46
ACSS2 Q9NR19 1/20 0.44
TSHR P16473 2/20 0.43
HSD17B10 Q99714 2/20 0.43
ACACB O00763 2/20 0.43
CNR2 P34972 1/20 0.43
BRD9 Q9H8M2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9709565 0.90 MEN1 (0.52) KDM4EMEN1KMT2AHTTGAA
SCHEMBL3924808 0.88 MEN1 (0.52) KDM4EMEN1KMT2AHTTGAA
SCHEMBL3924829 0.81 HTT (0.75) KDM4EMEN1KMT2AHTTGAA
SCHEMBL27837493 0.78 MEN1 (0.52) KDM4EMEN1KMT2AHTTGAA
SCHEMBL15919362 0.77 ACP1 (0.56) KDM4EMEN1KMT2AHTTGAA
SCHEMBL13742891 0.74 GAA (0.74) KDM4EMEN1KMT2AHTTGAA
SCHEMBL28499306 0.74 HTT (0.55) KDM4EMEN1KMT2AHTTGAA
SCHEMBL17981164 0.73 PTPN1 (0.56) KDM4EMEN1KMT2AHTTGAA
SCHEMBL17447717 0.73 MEN1 (0.53) KDM4EMEN1KMT2AHTTGAA
SCHEMBL5757395 0.72 POLB (0.47) ALDH1A1TSHRCNR2BRD9POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992022533-A1 4-AMINOQUINOLINES AND PHARMACEUTICAL COMPOSITIONS THEREOF THE UPJOHN COMPANY (US) 1992-12-23 WO disclosed