SCHEMBL9710209

SCHEMBL9710209

COc1ccc(C(N)=O)c(SSc2cc(OC)ccc2C(N)=O)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 1/20 0.49
PARP1 P09874 3/20 0.48
PARP10 Q53GL7 2/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
PARP2 Q9UGN5 1/20 0.48
PARP4 Q9UKK3 1/20 0.48
ALDH1A1 P00352 5/20 0.47
HPGD P15428 4/20 0.47
MAPK1 P28482 3/20 0.47
CYP3A4 P08684 2/20 0.47
RAD52 P43351 1/20 0.46
GAA P10253 2/20 0.44
CASP1 P29466 1/20 0.43
PLA2G10 O15496 1/20 0.43
LMNA P02545 2/20 0.42
CYP1A2 P05177 2/20 0.42
PGR P06401 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8379210 0.86 KDM4E (0.49) KDM4ENPC1RAB9APARP1PARP10
SCHEMBL11175864 0.84 ALDH1A1 (0.62) KDM4ENPC1RAB9AALDH1A1HPGD
SCHEMBL826392 0.84 SMN1; SMN2 (0.53) KDM4ENPC1RAB9ACA1CA2
SCHEMBL6225082 0.82 NPC1 (0.49) KDM4ENPC1RAB9AALDH1A1HPGD
SCHEMBL2835948 0.81 PARP1 (0.55) KDM4ENPC1RAB9APARP1PARP10
SCHEMBL1807116 0.79 PARP1 (0.53) KDM4ENPC1RAB9APARP1PARP10
SCHEMBL12264144 0.78 SMN1; SMN2 (0.51) KDM4ENPC1RAB9AALDH1A1HPGD
SCHEMBL3343162 0.78 PARP1 (0.52) KDM4ENPC1RAB9APARP1PARP10
SCHEMBL1034025 0.78 ALDH1A1 (0.68) NPC1RAB9APARP10CA1CA2
SCHEMBL1447373 0.78 NPC1 (0.72) KDM4ENPC1RAB9APARP1PARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992021668-A1 BENZOTHIAZEPINONES AND THEIR USE AS ANTICONVULSANTS THE BOOTS COMPANY PLC (GB) 1992-12-10 WO disclosed