SCHEMBL9710552

SCHEMBL9710552

CCc1[nH]c(=O)oc1-c1ccc(-n2ccnc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADH5 P11766 2/20 0.52
PDE4A P27815 5/20 0.52
PDE4B Q07343 5/20 0.52
PDE4C Q08493 5/20 0.52
PDE4D Q08499 5/20 0.52
PDE3B Q13370 10/20 0.47
PDE3A Q14432 10/20 0.47
PDE2A O00408 2/20 0.46
TSHR P16473 2/20 0.44
MEN1 O00255 1/20 0.44
ALOX15 P16050 1/20 0.44
KMT2A Q03164 1/20 0.44
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
LMNA P02545 1/20 0.43
MAPK1 P28482 1/20 0.43
PDE1A P54750 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7272043 0.78 PDE3B (0.43) PDE3BPDE3AKMT2ACYP1A2CYP2C19
SCHEMBL10756489 0.73 PDE3B (0.55) ADH5PDE4APDE4BPDE4CPDE4D
SCHEMBL10771601 0.70 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9705393 0.70 NOTUM (0.45) MEN1KMT2ACYP3A4
SCHEMBL2533488 0.69 TSHR (0.84) ADH5PDE4APDE4BPDE4CPDE4D
SCHEMBL8392834 0.69 MEN1 (0.61) ADH5PDE3BPDE3APDE2ATSHR
SCHEMBL7342584 0.68 PDE3B (0.49) ADH5PDE4APDE4BPDE4CPDE4D
SCHEMBL7266072 0.68 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL255498 0.68 MAOB (0.62) TSHRMEN1ALOX15KMT2ACYP1A2
SCHEMBL16568283 0.68 PDE3B (0.50) ADH5PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0223177-B1 CARDIOTONIC PHENYL OXAZOLONES MERRELL DOW PHARMACEUTICALS INC. (US) 1992-08-19 EP disclosed
US-4728661-A Cardiotonic phenyl oxazolones MERRELL DOW PHARMACEUTICALS INC. (US) 1988-03-01 US disclosed