SCHEMBL9711186

SCHEMBL9711186

O=C(S)Cc1c(F)c(F)cc(F)c1F

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
CA4 P22748 2/20 0.41
CES2 O00748 4/20 0.39
CES1 P23141 4/20 0.39
CA12 O43570 1/20 0.32
CA7 P43166 1/20 0.32
CA13 Q8N1Q1 1/20 0.32
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6858299 0.81 CA1 (0.44) CA1CA2CA4CES2CES1
SCHEMBL11269548 0.79 CA1 (0.43) CA1CA2CA4CES2CES1
SCHEMBL28207133 0.77 CA2 (0.41) CA1CA2CA4CES2CES1
SCHEMBL27110079 0.77 CA1 (0.41) CA1CA2CA4CES2CES1
SCHEMBL9711188 0.70 CA1 (0.33) CA1CA2CA4CES2CES1
SCHEMBL28231870 0.70 KDM4E (0.50) CES1MAPT
SCHEMBL6863804 0.68 CA1 (0.41) CA1CA2CA4CES2CES1
SCHEMBL20881848 0.68 CA1 (0.32) CA1CA2CA4CES2CES1
SCHEMBL1070979 0.67 CA1 (0.39) CA1CA2CA4CES2CES1
SCHEMBL358960 0.67 CA1 (0.39) CA1CA2CA4CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5153227-A Treatment of diabetes and galactosemia complications IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-10-06 US disclosed
EP-0304190-B1 (ARYLSULPHONYL)NITROMETHANES, PROCESS FOR THEIR PREPARATION AND USE IN PHARMACEUTICAL COMPOSITIONS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-07-08 EP disclosed
EP-0304190-A1 (Arylsulphonyl)nitromethanes, process for their preparation and use in pharmaceutical compositions IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-02-22 EP disclosed