SCHEMBL9714474

SCHEMBL9714474

COc1cc(C(=O)N(NC(=O)c2ccccc2)C(C)(C)C)ccc1[N+](=O)[O-]

nearest known ligand 0.64

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.60
CYP2C9 P11712 1/20 0.60
POLB P06746 1/20 0.57
ABCB1 P08183 2/20 0.48
ALDH1A1 P00352 1/20 0.47
TSHR P16473 1/20 0.47
TDP1 Q9NUW8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9714470 0.96 POLB (0.57) CYP3A4CYP2C9POLBABCB1ALDH1A1
SCHEMBL10749557 0.80 POLB (0.68) CYP3A4CYP2C9POLBABCB1ALDH1A1
SCHEMBL9825776 0.80 POLB (0.68) CYP3A4CYP2C9POLBABCB1
SCHEMBL9714603 0.79 CYP3A4 (0.73) CYP3A4CYP2C9POLBABCB1
SCHEMBL9714499 0.79 ABCB1 (0.57) CYP3A4CYP2C9POLBABCB1
SCHEMBL9557393 0.79 ALDH1A1 (0.43) CYP3A4ABCB1ALDH1A1TSHRTDP1
SCHEMBL8166763 0.79 POLB (0.74) CYP3A4CYP2C9POLBABCB1
SCHEMBL9652010 0.79 POLB (0.74) CYP3A4CYP2C9POLBABCB1
SCHEMBL9714310 0.78 POLB (0.68) CYP3A4CYP2C9POLBABCB1
SCHEMBL9825764 0.78 POLB (0.68) CYP3A4CYP2C9POLBABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0245950-B1 INSECTICIDAL N-SUBSTITUTED-N' - SUBSTITUTED-N, N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1992-06-17 EP disclosed
EP-0236618-B1 INSECTICIDAL N'-SUBSTITUTED-N,N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1991-02-27 EP disclosed
US-4985461-A Insecticidal N'-substituted-N,N'-diacylhydrazines ROHM AND HAAS COMPANY (US) 1991-01-15 US disclosed
EP-0236618-A2 Insecticidal N'-substituted-N,N'-diacylhydrazines ROHM AND HAAS COMPANY (US) 1987-09-16 EP disclosed