SCHEMBL9717852

SCHEMBL9717852

C[C@H](N)C(=O)c1nc(C[C@H](N)C(=O)O)c[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.43
SLC7A5 Q01650 3/20 0.41
CYP3A4 P08684 3/20 0.41
KDM4E B2RXH2 3/20 0.38
LMNA P02545 3/20 0.38
MAPT P10636 3/20 0.38
BLM P54132 3/20 0.38
PMP22 Q01453 3/20 0.38
KMT2A Q03164 3/20 0.38
TSHR P16473 2/20 0.38
MEN1 O00255 2/20 0.38
HIF1A Q16665 2/20 0.38
MPO P05164 1/20 0.38
PKM P14618 2/20 0.37
ALPI P09923 1/20 0.37
PTGS1 P23219 1/20 0.37
XIAP P98170 1/20 0.37
GRIA2 P42262 4/20 0.35
GRIA1 P42261 3/20 0.35
GRIA3 P42263 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9717841 1.00 CYP1A2 (0.43) CYP1A2SLC7A5CYP3A4KDM4ELMNA
SCHEMBL359889 0.84 CYP1A2 (0.42) CYP1A2SLC7A5CYP3A4KDM4ELMNA
SCHEMBL31370049 0.83 CYP1A2 (0.46) CYP1A2SLC7A5CYP3A4KDM4ELMNA
SCHEMBL25354300 0.82 CYP1A2 (0.43) CYP1A2SLC7A5CYP3A4KDM4ELMNA
SCHEMBL25354296 0.82 CYP1A2 (0.43) CYP1A2SLC7A5CYP3A4KDM4ELMNA
SCHEMBL25354014 0.81 SLC7A5 (0.44) CYP1A2SLC7A5CYP3A4KDM4ELMNA
SCHEMBL25354020 0.81 SLC7A5 (0.44) CYP1A2SLC7A5CYP3A4KDM4ELMNA
SCHEMBL31295696 0.80 CYP1A2 (0.41) CYP1A2SLC7A5CYP3A4KDM4ELMNA
SCHEMBL7782852 0.79 CYP1A2 (0.43) CYP1A2SLC7A5CYP3A4KDM4ELMNA
SCHEMBL31369922 0.79 SLC7A5 (0.43) CYP1A2SLC7A5CYP3A4KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0436611-A4 COMPOUND AND METHOD FOR THE RETARDATION OF COLLAGEN CROSS-LINKING 1992-03-11 EP disclosed
EP-0436611-A1 COMPOUND AND METHOD FOR THE RETARDATION OF COLLAGEN CROSS-LINKING COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 1991-07-17 EP disclosed
WO-1990006102-A1 COMPOUND AND METHOD FOR THE RETARDATION OF COLLAGEN CROSS-LINKING PEPTIDE TECHNOLOGY LIMITED (AU) 1990-06-14 WO disclosed