SCHEMBL9720561

SCHEMBL9720561

CCC(=O)c1c(C)cc(Cl)cc1C

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
PTGS1 P23219 1/20 0.47
DRD3 P35462 1/20 0.47
ALOX15 P16050 1/20 0.41
TSHR P16473 2/20 0.41
SMN1; SMN2 Q16637 3/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPK1 P28482 1/20 0.38
POLB P06746 2/20 0.37
ABCB1 P08183 1/20 0.37
THRB P10828 2/20 0.36
THRA P10827 1/20 0.36
RAB9A P51151 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
KDM4E B2RXH2 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11210247 0.82 MEN1 (0.50) CYP3A4MEN1KMT2APTGS1DRD3
SCHEMBL2380078 0.81 GSK3B (0.45) MEN1KMT2ASMN1; SMN2ALDH1A1MAPK1
SCHEMBL28155500 0.80 CYP3A4 (0.65) CYP3A4MEN1KMT2APTGS1DRD3
SCHEMBL11217214 0.80 KMT2A (0.48) CYP3A4MEN1KMT2APTGS1DRD3
SCHEMBL9634983 0.78 KMT2A (0.47) CYP3A4MEN1KMT2APTGS1DRD3
SCHEMBL28091418 0.78 CYP3A4 (0.47) CYP3A4MEN1KMT2APTGS1DRD3
SCHEMBL29059825 0.77 MEN1 (0.45) CYP3A4MEN1KMT2APTGS1DRD3
SCHEMBL27788907 0.77 TSHR (0.46) CYP3A4MEN1KMT2APTGS1DRD3
SCHEMBL9720612 0.75 CYP3A4 (0.57) CYP3A4MEN1KMT2APTGS1DRD3
SCHEMBL13545162 0.75 KMT2A (0.44) CYP3A4MEN1KMT2APTGS1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105906617-A Modulators of HEC1 activity and methods thereof 泰纬生命科技股份有限公司 2016-08-31 CN disclosed
US-5103022-A Reacting dl-2-methyl-1-(4-trifluoromethylphenyl)-3-pyrrolidino -1-propanone with l-acetylphenylglycine to form corresponding diastereomeric salt, deposition, isolation of l-2-methyl-1-(4-trifluoromethylphenyl)-3-pyrrolidino-1-propanone NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1992-04-07 US disclosed
US-5057535-A Muscle relaxants NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1991-10-15 US disclosed
EP-0200942-A2 New derivatives of an aminoketone NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1986-11-12 EP disclosed