SCHEMBL27788907

SCHEMBL27788907

CCC(=O)c1c(F)cc(Cl)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.46
KMT2A Q03164 4/20 0.45
MEN1 O00255 3/20 0.45
CYP3A4 P08684 2/20 0.45
PTGS1 P23219 1/20 0.45
DRD3 P35462 1/20 0.45
ALOX15 P16050 1/20 0.37
KCNH2 Q12809 1/20 0.36
CCNB2 O95067 1/20 0.36
CCNE2 O96020 1/20 0.36
CDK1 P06493 1/20 0.36
CDK4 P11802 1/20 0.36
CCNB1 P14635 1/20 0.36
CCND1 P24385 1/20 0.36
CCNE1 P24864 1/20 0.36
CDK2 P24941 1/20 0.36
CCND2 P30279 1/20 0.36
CCND3 P30281 1/20 0.36
CCNB3 Q8WWL7 1/20 0.36
MAPT P10636 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27789001 0.89 MEN1 (0.53) TSHRKMT2AMEN1CYP3A4PTGS1
SCHEMBL3422296 0.83 KMT2A (0.48) TSHRKMT2AMEN1CYP3A4PTGS1
SCHEMBL16284311 0.81 CYP3A4 (0.63) TSHRKMT2AMEN1CYP3A4PTGS1
SCHEMBL29924838 0.81 GSK3B (0.43) KMT2AMEN1MAPTALDH1A1SMN1; SMN2
SCHEMBL28080415 0.79 MEN1 (0.45) TSHRKMT2AMEN1CYP3A4PTGS1
SCHEMBL27841431 0.79 MEN1 (0.45) TSHRKMT2AMEN1CYP3A4PTGS1
SCHEMBL11217214 0.78 KMT2A (0.48) TSHRKMT2AMEN1CYP3A4PTGS1
SCHEMBL9720561 0.77 CYP3A4 (0.47) TSHRKMT2AMEN1CYP3A4PTGS1
SCHEMBL28091408 0.76 KMT2A (0.49) KMT2AMEN1CYP3A4PTGS1DRD3
SCHEMBL28174203 0.76 TSHR (0.47) TSHRKMT2AMEN1CYP3A4PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101809005-B Fused bicyclic compound MITSUBISHI TANABE PHARMA CORP 2013-05-01 CN disclosed
CN-101809005-A Fused bicyclic compound MITSUBISHI TANABE PHARMA CORP 2010-08-18 CN disclosed