SCHEMBL9720896

SCHEMBL9720896

CN1C(=O)CN(CCCN2CC(=O)N(C)C(=O)C2)CC1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.38
DRD2 P14416 2/20 0.37
HTR7 P34969 2/20 0.37
HTR1A P08908 1/20 0.37
HTR2C P28335 1/20 0.37
HRH1 P35367 1/20 0.37
HTR2B P41595 1/20 0.37
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
NFKB1 P19838 1/20 0.33
PTGS1 P23219 1/20 0.33
APEX1 P27695 1/20 0.33
THPO P40225 1/20 0.33
PMP22 Q01453 1/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3333138 0.89 PIK3CD (0.40) PIK3CDDRD2HTR7HTR1AHTR2C
SCHEMBL12208456 0.79 PIK3CD (0.38) PIK3CDMEN1LMNACYP3A4CYP2C9
SCHEMBL15549868 0.77 PIK3CD (0.36) PIK3CDMEN1LMNACYP3A4CYP2C9
SCHEMBL15548788 0.72 TSHR (0.39) PIK3CDMEN1LMNACYP3A4CYP2C9
SCHEMBL84388 0.71 GSK3A (0.35) PTGS1GSK3AGSK3B
SCHEMBL9720830 0.69 PTGS1 (0.56) PIK3CDMEN1LMNACYP3A4CYP2C9
SCHEMBL9720746 0.69 PTGS1 (0.56) PIK3CDMEN1LMNACYP3A4CYP2C9
SCHEMBL9720744 0.69 PTGS1 (0.56) PIK3CDMEN1LMNACYP3A4CYP2C9
SCHEMBL9752550 0.68 TOP2A (0.47) DRD2HTR7HTR1AHTR2CHRH1
SCHEMBL1101974 0.68 MC4R (0.53) MEN1LMNAKMT2AALDH1A1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992000740-A2 BIS-DIOXOPIPERAZINES AND THEIR USE AS PROTECTION AGENTS NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1992-01-23 WO disclosed