SCHEMBL9752550

SCHEMBL9752550

O=C1CN(CCCN2CC(=O)NC(=O)C2)CC(=O)N1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 3/20 0.47
TOP2B Q02880 3/20 0.47
PTGS1 P23219 2/20 0.47
LMNA P02545 2/20 0.47
CRBN Q96SW2 3/20 0.44
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
HTR2C P28335 1/20 0.33
HTR7 P34969 1/20 0.33
HRH1 P35367 1/20 0.33
HTR2B P41595 1/20 0.33
CXCR4 P61073 1/20 0.32
SIGMAR1 Q99720 3/20 0.32
USP2 O75604 1/20 0.31
POLB P06746 1/20 0.31
ALOX15 P16050 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL728996 0.89 TOP2A (0.50) TOP2ATOP2BPTGS1LMNACRBN
SCHEMBL11383117 0.86 PTGS1 (0.46) TOP2ATOP2BPTGS1LMNACRBN
SCHEMBL11023978 0.84 ALDH1A1 (0.47) TOP2ATOP2BPTGS1LMNACRBN
SCHEMBL5707893 0.80 TOP2A (0.48) TOP2ATOP2BPTGS1LMNACRBN
SCHEMBL29130872 0.80 PTGS1 (0.44) TOP2ATOP2BPTGS1LMNACRBN
SCHEMBL16876983 0.80 PTGS1 (0.37) TOP2ATOP2BPTGS1LMNACRBN
SCHEMBL31377154 0.75 APEX1 (0.42) TOP2ATOP2BPTGS1LMNACRBN
SCHEMBL1101973 0.75
SCHEMBL15548784 0.74 TOP2A (0.47) TOP2ATOP2BPTGS1LMNACRBN
SCHEMBL16349791 0.74 TOP2A (0.52) TOP2ATOP2BPTGS1LMNACRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991000729-A2 BIS-DIOXOPIPERAZINES, AND THEIR USE AS PROTECTING AGENTS NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1991-01-24 WO disclosed
EP-0409499-A2 Pharmaceutical compositions BTG INTERNATIONAL LIMITED (GB) 1991-01-23 EP disclosed
EP-0408384-A1 N,N'-dicarboxymethyl, N,N'-dicarbamoylmethyl diaminoalkane derivatives and their use in pharmaceutical compositions. BTG INTERNATIONAL LIMITED (GB) 1991-01-16 EP disclosed