SCHEMBL9722601

SCHEMBL9722601

C=C1/C(=C\C=C2CCC[C@@]3(C)C2CC[C@@H]3[C@H](C)CCC[C@](C)(O)CO)C[C@@H](O)C[C@H]1O

nearest known ligand 0.86

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VDR P11473 11/20 0.86
MAPT P10636 3/20 0.86
ADORA3 P0DMS8 2/20 0.86
SLC6A2 P23975 2/20 0.86
AGTR1 P30556 2/20 0.86
SMN1; SMN2 Q16637 2/20 0.86
NR1I2 O75469 1/20 0.86
ABCB11 O95342 1/20 0.86
GC P02774 1/20 0.86
PGR P06401 1/20 0.86
RXRA P19793 1/20 0.86
CHRM3 P20309 1/20 0.86
CNR1 P21554 1/20 0.86
HTR2C P28335 1/20 0.86
MAPK1 P28482 1/20 0.86
SLC6A4 P31645 1/20 0.86
ADRA1A P35348 1/20 0.86
PTGS2 P35354 1/20 0.86
OPRD1 P41143 1/20 0.86
OPRK1 P41145 1/20 0.86

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9722585 1.00 VDR (0.86) VDRMAPTADORA3SLC6A2AGTR1
SCHEMBL10445242 1.00 VDR (0.86) VDRMAPTADORA3SLC6A2AGTR1
SCHEMBL11165113 1.00 VDR (0.86) VDRMAPTADORA3SLC6A2AGTR1
SCHEMBL10892411 1.00 VDR (0.86) VDRMAPTADORA3SLC6A2AGTR1
SCHEMBL10895773 1.00 VDR (0.86) VDRMAPTADORA3SLC6A2AGTR1
SCHEMBL23359068 1.00 VDR (0.86) VDRMAPTADORA3SLC6A2AGTR1
SCHEMBL9722594 1.00 VDR (0.86) VDRMAPTADORA3SLC6A2AGTR1
SCHEMBL9173699 1.00 VDR (0.86) VDRMAPTADORA3SLC6A2AGTR1
SCHEMBL9722605 1.00 VDR (0.86) VDRMAPTADORA3SLC6A2AGTR1
SCHEMBL10892402 1.00 VDR (0.86) VDRMAPTADORA3SLC6A2AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-58210017-A None JP disclosed
WO-2023068322-A1 CD RING SIDE CHAIN-SUBSTITUTED VITAMIN D DERIVATIVE 学校法人帝京大学 2023-04-27 WO disclosed
US-5120722-A Trihydroxy-cholecacliferol and trihydroxy-ergocalciferol for treating leukemia HOFFMANN-LA ROCHE INC. (US) 1992-06-09 US disclosed
US-5110958-A Antitumor agents HOFFMANN-LA ROCHE INC. (US) 1992-05-05 US disclosed
EP-0154185-B1 CALCIFEROL DERIVATIVES F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1988-10-05 EP disclosed
US-4749710-A HYDROXYLATED ERGOCALCIFEROLS; ADMINISTERING HOFFMANN-LA ROCHE INC. (US) 1988-06-07 US disclosed
US-4617297-A CALCIUM METABOLIC DISORDERS HOFFMANN-LA ROCHE INC. (US) 1986-10-14 US disclosed
JP-S58210017-A ANTITUMOR AGENT KUREHA CHEM IND CO LTD 1983-12-07 JP disclosed