SCHEMBL9722609

SCHEMBL9722609

O=C(CNc1ccccn1)CNc1ccccn1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.58
NPC1 O15118 5/20 0.57
RAB9A P51151 5/20 0.57
PKM P14618 2/20 0.57
CXCR4 P61073 1/20 0.55
FABP1 P07148 1/20 0.53
FABP6 P51161 1/20 0.53
FDPS P14324 1/20 0.53
ALDH1A1 P00352 1/20 0.51
HPGD P15428 1/20 0.51
CYP2D6 P10635 1/20 0.50
CYP1A2 P05177 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
CYP2C19 P33261 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
PIM1 P11309 1/20 0.49
ADORA2A P29274 1/20 0.49
ADORA2B P29275 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL534155 0.86 GAA (0.56) GAANPC1RAB9APKMCXCR4
Hydrochloric Acid SCHEMBL360682 0.86 GAA (0.56) GAANPC1RAB9APKMCXCR4
SCHEMBL13589538 0.85 GAA (0.55) GAANPC1RAB9APKMCXCR4
SCHEMBL2857962 0.85 GAA (0.55) GAANPC1RAB9APKMCXCR4
SCHEMBL28664986 0.83 GAA (0.53) GAANPC1RAB9APKMCXCR4
SCHEMBL28643003 0.82 GAA (0.56) GAANPC1RAB9APKMCXCR4
SCHEMBL22338218 0.82 GAA (0.56) GAANPC1RAB9APKMCXCR4
SCHEMBL7436411 0.82 GAA (0.51) GAANPC1RAB9APKMCXCR4
SCHEMBL15785585 0.81
Hydrochloric Acid SCHEMBL7494264 0.80 GAA (0.50) GAANPC1RAB9APKMCXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5106986-A PREPARATION OF AMINOETHANOL DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 1992-04-21 US claimed
EP-0450180-A2 Process for the preparation of aminoethanol derivatives BAYER AG (DE) 1991-10-09 EP claimed
JP-4211658-A None JP disclosed
JP-H04211658-A PREPARATION OF AMINOETHANOL DERIVATIVE BAYER AG 1992-08-03 JP disclosed
US-5106986-A PREPARATION OF AMINOETHANOL DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 1992-04-21 US disclosed
EP-0450180-A2 Process for the preparation of aminoethanol derivatives BAYER AG (DE) 1991-10-09 EP disclosed
EP-0450180-A2 Process for the preparation of aminoethanol derivatives BAYER AG (DE) 1991-10-09 EP disclosed
US-4895950-A 5-halogeno-6-amino-nicotinic acid halides BAYER AKTIENGESELLSCHAFT (DE) 1990-01-23 US disclosed
EP-0302227-A2 5-Halo-6-amino-nicotinic acid halides, their preparation and their use BAYER AG (DE) 1989-02-08 EP disclosed