SCHEMBL9722753

SCHEMBL9722753

COC(=O)c1cccc2sc(N)nc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
ALDH1A1 P00352 8/20 0.53
PDPK1 O15530 1/20 0.53
GAA P10253 4/20 0.49
MAPK1 P28482 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
LMNA P02545 1/20 0.49
PDE10A Q9Y233 1/20 0.49
HSD17B10 Q99714 3/20 0.47
CFTR P13569 1/20 0.47
KDM4E B2RXH2 5/20 0.47
HPGD P15428 3/20 0.47
MAPT P10636 5/20 0.46
PPARG P37231 1/20 0.46
NCOA2 Q15596 1/20 0.46
NCOA1 Q15788 1/20 0.46
NCOA3 Q9Y6Q9 1/20 0.46
KMT2A Q03164 3/20 0.45
ATM Q13315 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9722823 0.84 ALDH1A1 (0.53) CYP3A4TDP1ALDH1A1PDPK1GAA
SCHEMBL2793048 0.84 ALDH1A1 (0.49) CYP3A4TDP1ALDH1A1PDPK1GAA
SCHEMBL12109867 0.83 MAPT (0.50) ALDH1A1GAAMAPK1LMNAHSD17B10
SCHEMBL1936413 0.82 ALDH1A1 (0.56) ALDH1A1GAASMN1; SMN2LMNAHSD17B10
SCHEMBL4470820 0.81 PDPK1 (0.59) CYP3A4TDP1ALDH1A1PDPK1SMN1; SMN2
SCHEMBL5670201 0.81 PDPK1 (0.59) CYP3A4TDP1ALDH1A1PDPK1GAA
SCHEMBL6477475 0.81 ALDH1A1 (0.45) CYP3A4TDP1ALDH1A1PDPK1GAA
Bromide SCHEMBL5669202 0.80 PDPK1 (0.57) CYP3A4TDP1ALDH1A1PDPK1GAA
SCHEMBL9619834 0.78 HSD17B10 (0.55) CYP3A4ALDH1A1GAAMAPK1SMN1; SMN2
SCHEMBL6057635 0.77 NSD1 (0.55) CYP3A4TDP1ALDH1A1GAAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120872-A Textile dyeing CIBA-GEIGY CORPORATION (US) 1992-06-09 US disclosed
US-4994563-A Dyeing, printing cellulose, silk, wool, synthetic polyamides; colorfastness CIBA-GEIGY CORPORATION (US) 1991-02-19 US disclosed
EP-0349486-A2 Azo dyes, their preparation and their use CIBA-GEIGY AG (CH) 1990-01-03 EP disclosed