SCHEMBL9724178

SCHEMBL9724178

C#CCNc1ccc(C(=O)N[C@H](CCC(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c(F)c1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TYMS P04818 4/20 0.38
DHFR P00374 1/20 0.38
GART P22102 1/20 0.37
KDR P35968 3/20 0.35
P2RY12 Q9H244 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9724176 1.00 TYMS (0.38) TYMSDHFRGARTKDRP2RY12
SCHEMBL6885924 0.87 TYMS (0.37) TYMSDHFRGARTKDRP2RY12
SCHEMBL6885928 0.87 TYMS (0.37) TYMSDHFRGARTKDRP2RY12
SCHEMBL9379559 0.84 L3MBTL1 (0.47) TYMSDHFRGART
SCHEMBL9379564 0.84 L3MBTL1 (0.47) TYMSDHFRGART
SCHEMBL6885646 0.84 POLB (0.41) TYMSDHFRGARTTDP1CYP3A4
SCHEMBL6885650 0.84 POLB (0.41) TYMSDHFRGARTTDP1CYP3A4
SCHEMBL9556071 0.84 P2RY12 (0.39) P2RY12TDP1
SCHEMBL9556079 0.84 P2RY12 (0.39) P2RY12TDP1
SCHEMBL15686202 0.82 P2RY12 (0.37) P2RY12TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed