SCHEMBL9724255

SCHEMBL9724255

Cc1ccc2nc(N)cc(C)c2c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.63
NCK1 P16333 1/20 0.55
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
ACHE P22303 5/20 0.50
BCHE P06276 4/20 0.50
GRIN1 Q05586 4/20 0.50
GRIN2A Q12879 4/20 0.50
LMNA P02545 2/20 0.47
GAA P10253 1/20 0.45
HTT P42858 1/20 0.45
ELANE P08246 1/20 0.44
PRMT5 O14744 1/20 0.44
NOS3 P29474 1/20 0.44
NOS1 P29475 1/20 0.44
NOS2 P35228 1/20 0.44
RAD52 P43351 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HRH4 Q9H3N8 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5456804 0.84 BACE1 (0.55) BACE1NCK1ACHEBCHEGRIN1
SCHEMBL11399020 0.81 BACE1 (0.52) BACE1NCK1MEN1KMT2AACHE
SCHEMBL17827033 0.81 LMNA (0.68) BACE1NCK1ACHEBCHEGRIN1
SCHEMBL3531515 0.79 LMNA (0.66) MEN1KMT2AACHEBCHEGRIN1
SCHEMBL11130296 0.78 BACE1 (0.56) BACE1MEN1KMT2ALMNAGAA
SCHEMBL9381975 0.78 BACE1 (0.49) BACE1NCK1MEN1KMT2AACHE
SCHEMBL3094768 0.78 BACE1 (1.00) BACE1ACHELMNAGAAPRMT5
SCHEMBL23757101 0.77 BACE1 (0.54) BACE1MEN1KMT2AGAAHTT
SCHEMBL2538787 0.76 KDM4E (0.66) MEN1KMT2AACHEBCHEGRIN1
SCHEMBL934670 0.76 KMT2A (0.56) MEN1KMT2AACHEBCHEGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed
EP-0318225-A2 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-31 EP disclosed