SCHEMBL9724271

SCHEMBL9724271

C#CCN(Cc1ccc2nc(C)cc(Br)c2c1)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)c(F)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
TYMS P04818 12/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9724187 0.91 TYMS (0.75) TYMS
SCHEMBL9556260 0.86 TYMS (1.00) TYMS
SCHEMBL9724196 0.85 TYMS (0.73) TYMS
SCHEMBL9724174 0.84 TYMS (0.75) TYMS
SCHEMBL9600838 0.82 TYMS (1.00) TYMS
SCHEMBL9724140 0.82 TYMS (0.68) TYMS
SCHEMBL9724111 0.82 TYMS (0.74) TYMS
SCHEMBL9724189 0.81 TYMS (0.72) TYMS
SCHEMBL9724165 0.81 TYMS (0.71) TYMS
SCHEMBL10828922 0.79 TYMS (0.74) TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed