SCHEMBL9724274

SCHEMBL9724274

O=CNC=Cc1ccc2ccccc2c1O

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.45
EGFR P00533 2/20 0.45
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
PKM P14618 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
CYP1B1 Q16678 6/20 0.43
ABCG2 Q9UNQ0 1/20 0.43
PTPN22 Q9Y2R2 1/20 0.43
MTNR1A P48039 1/20 0.42
MTNR1B P49286 1/20 0.42
CYP1A1 P04798 4/20 0.41
LDHA P00338 1/20 0.41
ERN1 O75460 1/20 0.41
NPC1 O15118 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9730667 0.78 ERN1 (0.46) KDM4EEGFRALDH1A1POLBGAA
SCHEMBL9731164 0.77 ERN1 (0.62) KDM4EEGFRALDH1A1POLBGAA
SCHEMBL9731169 0.77 ERN1 (0.62) KDM4EEGFRALDH1A1POLBGAA
SCHEMBL9731127 0.77 EGFR (0.53) KDM4EEGFRALDH1A1POLBGAA
SCHEMBL589343 0.77 ERN1 (0.55) ALDH1A1MAPTCYP1B1PTPN22CYP1A1
SCHEMBL9732410 0.77 EGFR (0.56) KDM4EEGFRALDH1A1POLBGAA
SCHEMBL9732522 0.76 EGFR (0.55) KDM4EEGFRALDH1A1POLBGAA
SCHEMBL8423542 0.76 CYP1B1 (0.55) KDM4EPKMCYP1B1ABCG2PTPN22
SCHEMBL8423545 0.76 CYP1B1 (0.55) KDM4EPKMCYP1B1ABCG2PTPN22
SCHEMBL9731055 0.75 EGFR (0.45) KDM4EEGFRALDH1A1POLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5122537-A Tyrosine kinase inhibitors FARMITALIA CARLO ERBA S.R.L. (IT) 1992-06-16 US claimed
JP-4210946-A None JP disclosed
JP-H04210946-A NEW ARYLVINYLAMIDE DERIVATIVE AND ITS PREPARATION FARMITALIA CARLO ERBA SPA 1992-08-03 JP disclosed
US-5122537-A Tyrosine kinase inhibitors FARMITALIA CARLO ERBA S.R.L. (IT) 1992-06-16 US disclosed