SCHEMBL9724344

SCHEMBL9724344

CC(=O)Nc1cc(C)c2cc(CBr)ccc2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.45
KDM4E B2RXH2 5/20 0.41
CYP2C19 P33261 2/20 0.41
CYP3A4 P08684 1/20 0.41
HIF1A Q16665 1/20 0.41
ALDH1A1 P00352 3/20 0.40
LMNA P02545 5/20 0.39
HPGD P15428 3/20 0.39
CYP2C9 P11712 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
GLA P06280 1/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
HSD17B10 Q99714 1/20 0.39
NPC1 O15118 1/20 0.39
ADORA3 P0DMS8 3/20 0.39
ADORA1 P30542 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ADORA2B P29275 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18317035 0.89 MEN1 (0.41) MAPTKDM4EALDH1A1LMNAHPGD
SCHEMBL9383680 0.85 NPC1 (0.41) MAPTKDM4EALDH1A1LMNAHPGD
SCHEMBL9724282 0.81 KMT2A (0.57) MAPTKDM4ECYP3A4ALDH1A1LMNA
SCHEMBL16930401 0.79 NPC1 (0.43) MAPTKDM4ECYP2C19CYP3A4LMNA
SCHEMBL16930398 0.77 NPC1 (0.44) MAPTKDM4ELMNASMN1; SMN2GLA
SCHEMBL16984472 0.77 KDM4E (0.55) MAPTKDM4EALDH1A1LMNAHPGD
SCHEMBL18325645 0.77 NPC1 (0.45) MAPTKDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL18317027 0.77 MEN1 (0.41) MAPTKDM4EALDH1A1LMNAHPGD
SCHEMBL18317003 0.76 MEN1 (0.43) MAPTKDM4EALDH1A1LMNAHPGD
Acetic Acid SCHEMBL9849558 0.76 KDM4E (0.54) MAPTKDM4EALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed
EP-0318225-A2 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-31 EP disclosed