SCHEMBL9724282

SCHEMBL9724282

CC(=O)Nc1cc(C)c2cc(C)ccc2n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.57
MEN1 O00255 2/20 0.57
ADORA3 P0DMS8 4/20 0.49
DYRK1A Q13627 2/20 0.49
GAA P10253 2/20 0.48
HTT P42858 2/20 0.48
ALDH1A1 P00352 4/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
ALOX15 P16050 1/20 0.46
KDM4E B2RXH2 4/20 0.46
LMNA P02545 2/20 0.45
NPC1 O15118 1/20 0.45
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.45
ADORA2A P29274 2/20 0.44
PKM P14618 1/20 0.44
ADORA1 P30542 2/20 0.43
ADORA2B P29275 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9724148 0.85 LMNA (0.55) KMT2AMEN1ADORA3DYRK1AHTT
SCHEMBL16984472 0.83 KDM4E (0.55) KMT2AMEN1ADORA3GAAALDH1A1
SCHEMBL9724344 0.81 MAPT (0.45) KMT2AMEN1ADORA3GAAALDH1A1
Acetic Acid SCHEMBL9849558 0.81 KDM4E (0.54) KMT2AMEN1ADORA3GAAALDH1A1
Potassium SCHEMBL30101822 0.81 KDM4E (0.54) KMT2AMEN1ADORA3GAAALDH1A1
SCHEMBL7056158 0.80 KMT2A (0.56) KMT2AMEN1GAAHTTALDH1A1
SCHEMBL15450991 0.78 DYRK1A (0.51) KMT2AMEN1ADORA3DYRK1AALDH1A1
SCHEMBL17646472 0.76 F2 (0.53) ADORA3DYRK1AHTTALDH1A1CYP1A2
SCHEMBL16930396 0.76 DYRK1A (0.53) KMT2AMEN1ADORA3DYRK1AALDH1A1
SCHEMBL7820537 0.75 ALDH1A1 (0.48) KMT2AMEN1ALDH1A1CYP1A2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed
EP-0318225-A2 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-31 EP disclosed