SCHEMBL9726532

SCHEMBL9726532

CCn1ncc(NCc2ccc(C)cc2C)c(C)c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 10/20 0.52
BRD9 Q9H8M2 9/20 0.52
NR3C1 P04150 1/20 0.45
PGR P06401 1/20 0.45
PDE4B Q07343 1/20 0.45
KAT2B Q92831 1/20 0.42
PKM P14618 1/20 0.40
PKLR P30613 1/20 0.40
BRPF1 P55201 1/20 0.40
BRD7 Q9NPI1 1/20 0.40
CNR2 P34972 1/20 0.39
P2RX7 Q99572 1/20 0.38
MAPT P10636 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
USP2 O75604 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
CASP1 P29466 1/20 0.37
HBB P68871 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10602234 0.88 BRD4 (0.54) BRD4BRD9NR3C1PGRPDE4B
SCHEMBL9726549 0.88 NR3C1 (0.44) BRD4BRD9NR3C1PGRPDE4B
SCHEMBL10602679 0.88 NR3C1 (0.44) BRD4BRD9NR3C1PGRPDE4B
SCHEMBL9726518 0.81 BRD4 (0.51) BRD4BRD9KAT2BBRPF1BRD7
SCHEMBL10601357 0.72 BRD4 (0.41) BRD4BRD9KAT2BPKMPKLR
SCHEMBL9726399 0.71 BRD4 (0.49) BRD4BRD9KAT2BMAPTGAA
SCHEMBL9726575 0.69 BRD4 (0.47) BRD4BRD9KAT2BBPTF
SCHEMBL9726418 0.69 KDM4E (0.46) BRD4BRD9MAPTKDM4EMEN1
SCHEMBL10601520 0.68 BRD4 (0.74) BRD4BRD9NR3C1KAT2BCNR2
SCHEMBL12497134 0.68 GAA (0.45) BRD4KAT2BMAPTMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098900-A Reducing contractions in smooth muscles NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1992-03-24 US disclosed
EP-0186817-B1 3(2H)PYRIDAZINONE, PROCESS FOR ITS PREPARATION AND ANTI-ALLERGIC AGENT CONTAINING IT NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1989-08-02 EP disclosed
EP-0186817-A1 3(2H)pyridazinone, process for its preparation and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1986-07-09 EP disclosed