SCHEMBL9726817

SCHEMBL9726817

Cc1ccc(C(=C(C=O)c2nnnn2C)c2ccc(C)cc2C)c(C)c1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
TP53 P04637 1/20 0.39
LMNA P02545 2/20 0.35
TSHR P16473 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
HMGCR P04035 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726768 0.88 HMGCR (0.36) ALDH1A1SMN1; SMN2NPC1RAB9ATP53
SCHEMBL9726524 0.88 HMGCR (0.36) ALDH1A1SMN1; SMN2NPC1RAB9ATP53
SCHEMBL9726571 0.87 HMGCR (0.35) ALDH1A1SMN1; SMN2NPC1RAB9ATP53
SCHEMBL9726576 0.87 HMGCR (0.41) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL9799375 0.79 SMN1; SMN2 (0.37) ALDH1A1SMN1; SMN2NPC1RAB9ATP53
SCHEMBL9799379 0.79 SMN1; SMN2 (0.37) ALDH1A1SMN1; SMN2NPC1RAB9ATP53
SCHEMBL9726563 0.77 HMGCR (0.44) HMGCR
SCHEMBL9726457 0.76 HMGCR (0.43) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL9726462 0.76 HMGCR (0.43) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL9726655 0.76 HMGCR (0.37) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US claimed
WO-1988006584-A1 ANTIHYPERCHOLESTEROLEMIC TETRAZOLE COMPOUNDS BRISTOL-MYERS COMPANY (US) 1988-09-07 WO claimed
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US disclosed
US-5068346-A Anticholesterol agents BRISTOL-MYERS COMPANY (US) 1991-11-26 US disclosed
US-4939265-A Intermediates and process for the preparation of antihypercholesterolemic tetrazole compounds BRISTOL-MYERS COMPANY (US) 1990-07-03 US disclosed
US-4898949-A Intermediates for the preparation of antihypercholesterolemic tetrazole compounds BRISTOL-MYERS COMPANY (US) 1990-02-06 US disclosed
US-4897490-A DERIVATIVES OF BETA-HYDROXY,OMEGA-DIPHENYL,TETRAZOL-5-YL ALK-OMEGA-ENOIC ACID, ESTER OR LACTONE BRISTOL-MEYERS COMPANY (US) 1990-01-30 US disclosed
WO-1988006584-A1 ANTIHYPERCHOLESTEROLEMIC TETRAZOLE COMPOUNDS BRISTOL-MYERS COMPANY (US) 1988-09-07 WO disclosed