SCHEMBL9726876

SCHEMBL9726876

COCCOCn1nnnc1C(C=CC(O)CC(O)CC(=O)O)=C(c1ccc(F)cc1)c1ccc(F)cc1

nearest known ligand 0.63

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 4/20 0.58
ESR1 P03372 1/20 0.40
CHRM1 P11229 1/20 0.40
TBXA2R P21731 1/20 0.40
PDE4A P27815 1/20 0.40
ADRA1A P35348 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726873 1.00 HMGCR (0.58) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9726976 0.92 HMGCR (0.70) HMGCR
SCHEMBL9726978 0.92 HMGCR (0.70) HMGCR
SCHEMBL9726991 0.86 HMGCR (0.65) HMGCR
SCHEMBL9726986 0.86 HMGCR (0.65) HMGCR
SCHEMBL10609441 0.84 HMGCR (0.49) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9726504 0.84 HMGCR (0.46) HMGCR
SCHEMBL9726497 0.84 HMGCR (0.46) HMGCR
SCHEMBL6258027 0.82 HMGCR (0.82) HMGCR
SCHEMBL9288114 0.82 HMGCR (0.82) HMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US disclosed
US-5068346-A Anticholesterol agents BRISTOL-MYERS COMPANY (US) 1991-11-26 US disclosed
US-4897490-A DERIVATIVES OF BETA-HYDROXY,OMEGA-DIPHENYL,TETRAZOL-5-YL ALK-OMEGA-ENOIC ACID, ESTER OR LACTONE BRISTOL-MEYERS COMPANY (US) 1990-01-30 US disclosed
WO-1988006584-A1 ANTIHYPERCHOLESTEROLEMIC TETRAZOLE COMPOUNDS BRISTOL-MYERS COMPANY (US) 1988-09-07 WO disclosed