SCHEMBL9728006

SCHEMBL9728006

CNc1ccc(C(C(C)C)n2ccnc2)cc1[N+](=O)[O-]

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 2/20 0.47
CYP19A1 P11511 2/20 0.45
CYP11B1 P15538 2/20 0.42
CYP11B2 P19099 2/20 0.42
HTT P42858 1/20 0.41
CYP26A1 O43174 7/20 0.41
CYP3A4 P08684 1/20 0.41
HCAR3 P49019 1/20 0.40
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fluorobenzene SCHEMBL10576700 0.92 CYP17A1 (0.48) CYP17A1CYP19A1CYP11B1CYP11B2HTT
SCHEMBL10580748 0.89 CYP19A1 (0.48) CYP17A1CYP19A1CYP11B1CYP11B2HTT
SCHEMBL10582410 0.87 MAPT (0.46) CYP17A1CYP19A1CYP11B1CYP11B2HTT
SCHEMBL9190551 0.83 CYP19A1 (0.50) CYP17A1CYP19A1CYP11B1CYP11B2CYP26A1
SCHEMBL10577494 0.83 CYP17A1 (0.48) CYP17A1CYP11B1CYP11B2HTTCYP3A4
SCHEMBL10581964 0.82 CYP19A1 (0.55) CYP17A1CYP19A1CYP11B1CYP11B2CYP26A1
SCHEMBL10698157 0.82 MAPT (0.46) CYP17A1CYP19A1HTTCYP26A1CYP3A4
SCHEMBL9728217 0.80 CYP17A1 (0.45) CYP17A1CYP11B1CYP11B2HTTCYP26A1
SCHEMBL9196029 0.80 L3MBTL1 (0.51) CYP17A1CYP11B1CYP11B2HTTCYP26A1
SCHEMBL9191000 0.80 CYP17A1 (0.44) CYP17A1CYP19A1CYP11B1CYP11B2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5151421-A Compounds for inhibition of metabolism of retinoids, for treatment for proliferation of epithelial cells and keratin disorders JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-29 US disclosed
US-5028606-A Retinoid metabolism inhibitors JANSSEN PHARMACEUTICA N.V. (BE) 1991-07-02 US disclosed
US-4859684-A (1H-imidazol-1-ylmethyl) substituted benzimidazole derivatives and use thereof in treating androgen dependent disorders JANSSEN PHARMACEUTICA N.V. (BE) 1989-08-22 US disclosed
EP-0260744-A2 (1H-imidazol-1-ylmethyl) substituted benzimidazole derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1988-03-23 EP disclosed