SCHEMBL9728136

SCHEMBL9728136

N#CN1C(=O)C(=O)c2ccccc21

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CES1 P23141 11/20 0.52
TTR P02766 1/20 0.52
BCHE P06276 4/20 0.50
TGM2 P21980 1/20 0.50
ALDH1A1 P00352 5/20 0.48
CES2 O00748 2/20 0.48
GAA P10253 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
ALDH3A1 P30838 4/20 0.44
ALDH2 P05091 3/20 0.44
CHRM1 P11229 2/20 0.44
CHRM5 P08912 1/20 0.44
CHRM3 P20309 1/20 0.44
PARK7 Q99497 1/20 0.42
ACHE P22303 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7300292 0.80 CES1 (0.57) CES1TTRBCHETGM2ALDH1A1
SCHEMBL30229556 0.77 CES1 (0.53) CES1TTRBCHETGM2ALDH1A1
SCHEMBL9550323 0.76 CA12 (0.43) ALDH1A1
SCHEMBL9143697 0.76 CA12 (0.43) ALDH1A1
SCHEMBL1749687 0.72 CES1 (0.57) CES1TTRBCHETGM2ALDH1A1
SCHEMBL31492057 0.72 CES1 (0.57) CES1TTRBCHETGM2ALDH1A1
SCHEMBL17818354 0.72 CES1 (0.57) CES1TTRBCHETGM2ALDH1A1
SCHEMBL31634050 0.72 CES1 (0.57) CES1TTRBCHETGM2ALDH1A1
SCHEMBL9179240 0.72 MAOA (0.70) CES1BCHETGM2ALDH1A1CES2
SCHEMBL27848668 0.72 CES1 (0.47) CES1TTRBCHETGM2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5151518-A N-arylation of isatins ABBOTT LABORATORIES (US) 1992-09-29 US disclosed