SCHEMBL9728160

SCHEMBL9728160

C=CCN(CC=C)C(=O)CN1CCCC1=O

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.51
POLB P06746 2/20 0.46
HTT P42858 1/20 0.42
ALDH1A1 P00352 2/20 0.41
BLM P54132 1/20 0.40
KMT2A Q03164 2/20 0.40
PIK3CD O00329 1/20 0.38
LMNA P02545 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5799328 0.79 TSHR (0.56) TSHRPOLBHTTALDH1A1KMT2A
SCHEMBL2036528 0.75 TSHR (0.59) TSHRPOLBHTTALDH1A1KMT2A
SCHEMBL16527290 0.74 HTT (0.55) TSHRPOLBHTTALDH1A1BLM
SCHEMBL11243429 0.72 TSHR (0.56) TSHRPOLBHTTALDH1A1KMT2A
SCHEMBL4372909 0.72 TSHR (0.51) TSHRPOLBHTTALDH1A1BLM
SCHEMBL10817574 0.72 TSHR (0.51) TSHRHTTALDH1A1BLMKMT2A
SCHEMBL1226609 0.71 TSHR (0.54) TSHRHTTALDH1A1BLMKMT2A
SCHEMBL917410 0.71 TSHR (0.58) TSHRHTTALDH1A1KMT2APIK3CD
SCHEMBL30762 0.70
SCHEMBL948990 0.70 TSHR (0.68) TSHRPOLBHTTALDH1A1BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175158-A CONDENSED DIAZEPINONES, PROCESSES FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS DR. KARL THOMAE, GMBH (DE) 1992-12-29 US disclosed
US-4931436-A BRADYCARDIAL AGENTS DR. KARL THOMAE GMBH (DE) 1990-06-05 US disclosed