SCHEMBL9728337

SCHEMBL9728337

CN(C)CCCC1CCCCN1CC(=O)N1c2ccccc2C(=O)Nc2cccnc21

nearest known ligand 0.85

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.75
CHRM4 P08173 3/20 0.75
CHRM1 P11229 3/20 0.75
CYP1A2 P05177 1/20 0.75
CYP3A4 P08684 1/20 0.75
CHRM3 P20309 1/20 0.75
MAPK1 P28482 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10514622 0.98 CHRM2 (0.74) CHRM2CHRM4CHRM1CYP1A2CYP3A4
SCHEMBL10508829 0.95 CHRM2 (0.77) CHRM2CHRM4CHRM1CYP1A2CYP3A4
SCHEMBL9727962 0.92 CHRM2 (0.83) CHRM2CHRM4CHRM1CYP1A2CYP3A4
SCHEMBL9597030 0.90 CYP1A2 (0.85) CHRM2CHRM4CHRM1CYP1A2CYP3A4
SCHEMBL9728148 0.90 CHRM2 (0.81) CHRM2CHRM4CHRM1CYP1A2CYP3A4
SCHEMBL10510299 0.89 CYP1A2 (0.85) CHRM2CHRM4CHRM1CYP1A2CYP3A4
SCHEMBL8881352 0.88 CHRM2 (0.71) CHRM2CHRM4CHRM1CYP1A2CYP3A4
SCHEMBL10515583 0.88 CYP1A2 (0.64) CHRM2CHRM4CHRM1CYP1A2CYP3A4
SCHEMBL9727602 0.87 CHRM2 (0.70) CHRM2CHRM4CHRM1CYP1A2CYP3A4
SCHEMBL9675477 0.87 CYP1A2 (0.58) CHRM2CHRM4CHRM1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175158-A CONDENSED DIAZEPINONES, PROCESSES FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS DR. KARL THOMAE, GMBH (DE) 1992-12-29 US disclosed
EP-0312895-A2 Condensed diazepinones, process for their preparation and medicament containing them Dr. Karl Thomae GmbH (DE) 1989-04-26 EP disclosed