SCHEMBL9729013

SCHEMBL9729013

NC(c1ccc(Br)cc1)c1ccccc1F

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.41
IDO1 P14902 2/20 0.41
TDO2 P48775 2/20 0.41
DPP4 P27487 1/20 0.39
GAA P10253 1/20 0.37
IGF1R P08069 1/20 0.36
HDAC4 P56524 4/20 0.34
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
MAPT P10636 2/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
NPC1 O15118 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
CNR1 P21554 1/20 0.33
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17842003 0.84 IDO1 (0.43) IDO1TDO2GAAHDAC4ALDH1A1
SCHEMBL3999911 0.84 IDO1 (0.55) IDO1TDO2DPP4GAACES2
SCHEMBL17842282 0.81 ADRB2 (0.42) IDO1TDO2GAAMEN1KMT2A
Hydrochloric Acid SCHEMBL32690499 0.79 IDO1 (0.43) IDO1TDO2GAAALDH1A1LMNA
SCHEMBL17842404 0.79 IDO1 (0.47) IDO1TDO2GAAMEN1KMT2A
SCHEMBL4505743 0.78 DPP4 (0.51) HTR2AIDO1TDO2DPP4KMT2A
SCHEMBL694825 0.77 IDO1 (0.41) IDO1TDO2GAAMEN1KMT2A
SCHEMBL16111744 0.77 HTR2A (0.37) HTR2AIDO1TDO2DPP4GAA
SCHEMBL16111990 0.77 IGF1R (0.42) HTR2AIDO1TDO2GAAIGF1R
SCHEMBL327420 0.76 IDO1 (0.51) HTR2AIDO1TDO2GAAIGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5081241-A Diabetes AMERICAN HOME PRODUCTS CORPORATION (US) 1992-01-14 US disclosed