SCHEMBL9730876

SCHEMBL9730876

CC(CN(C)C)C(=O)c1ccc2c(c1)OCC(=O)N2C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 2/20 0.41
CYP11B1 P15538 1/20 0.41
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
HTR1A P08908 3/20 0.37
HTR2C P28335 2/20 0.37
USP30 Q70CQ3 1/20 0.37
GABRA5 P31644 2/20 0.36
GABRA1 P14867 1/20 0.36
F10 P00742 1/20 0.36
EGFR P00533 1/20 0.35
CMA1 P23946 1/20 0.35
PTGER3 P43115 1/20 0.35
IDH1 O75874 1/20 0.35
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL9731026 0.83 CYP11B2 (0.41) CYP11B2CYP11B1PDE3BPDE3AHTR1A
SCHEMBL7343775 0.82 CYP11B2 (0.40) CYP11B2CYP11B1PDE3BPDE3AHTR1A
SCHEMBL21818855 0.77 CYP11B2 (0.50) CYP11B2CYP11B1PDE3BPDE3AHTR1A
SCHEMBL8146771 0.77 CYP11B2 (0.50) CYP11B2CYP11B1PDE3BPDE3AHTR1A
SCHEMBL9590395 0.75 MAPT (0.48) PDE3BPDE3AALDH1A1
SCHEMBL7485816 0.75 USP30 (0.46) CYP11B2CYP11B1PDE3BPDE3AUSP30
SCHEMBL474743 0.74 SMN1; SMN2 (0.53) CYP11B2CYP11B1PDE3BPDE3AHTR1A
SCHEMBL30040938 0.74 SMN1; SMN2 (0.53) CYP11B2CYP11B1PDE3BPDE3AHTR1A
SCHEMBL13409750 0.73 CYP11B2 (0.49) CYP11B2CYP11B1PDE3BPDE3AHTR1A
SCHEMBL7342699 0.73 USP30 (0.46) PDE3BPDE3AUSP30PTGER3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5081242-A Cardiotonic and bronchodilator agents; phosphodiesterase inhibitors ORTHO PHARMACEUTICAL CORPORATION (US) 1992-01-14 US claimed
EP-0272914-A2 6-Benzoxazinyl- and 6-benzothiazinyl-2,3,4,5-tetrahydropyridazin-3-ones ORTHO PHARMACEUTICAL CORPORATION (US) 1988-06-29 EP claimed