SCHEMBL9731015

SCHEMBL9731015

CCC1COC(c2ccc(-c3ccc(F)cc3)nc2)OC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 1/20 0.40
KDM1A O60341 10/20 0.38
NPC1 O15118 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
AURKA O14965 1/20 0.37
ABL1 P00519 1/20 0.37
NTRK1 P04629 1/20 0.37
LCK P06239 1/20 0.37
CSF1R P07333 1/20 0.37
RET P07949 1/20 0.37
MET P08581 1/20 0.37
PDGFRB P09619 1/20 0.37
PIM1 P11309 1/20 0.37
PDGFRA P16234 1/20 0.37
FLT3 P36888 1/20 0.37
MAPK8 P45983 1/20 0.37
CDK8 P49336 1/20 0.37
MAP2K1 Q02750 1/20 0.37
MAP4K2 Q12851 1/20 0.37
ROCK1 Q13464 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9365099 1.00 GRIA2 (0.40) GRIA2KDM1ANPC1RXFP1AURKA
SCHEMBL9366626 0.90 GRIA2 (0.39) GRIA2KDM1ANPC1RXFP1AURKA
SCHEMBL9366634 0.90 GRIA2 (0.39) GRIA2KDM1ANPC1RXFP1AURKA
SCHEMBL9366591 0.88 GRIA2 (0.38) GRIA2KDM1ANPC1RXFP1AURKA
SCHEMBL9366580 0.88 GRIA2 (0.38) GRIA2KDM1ANPC1RXFP1AURKA
SCHEMBL9370824 0.87 KDM1A (0.50) KDM1AMAOBGRM5DGAT1
SCHEMBL9366265 0.87 GRIA2 (0.37) GRIA2KDM1ANPC1RXFP1AURKA
SCHEMBL9366256 0.87 GRIA2 (0.37) GRIA2KDM1ANPC1RXFP1AURKA
SCHEMBL9366501 0.86 GRM2 (0.43) KDM1ANPC1MAOBCYP11B1CYP11B2
SCHEMBL9731106 0.86 GRM2 (0.43) KDM1ANPC1MAOBCYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5160661-A DIOXANYLPYRIDINE HOFFMANN-LA ROCHE INC. (US) 1992-11-03 US disclosed