SCHEMBL9732504

SCHEMBL9732504

O=CC1Cc2ccccc2C(=O)N1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.59
CA12 O43570 1/20 0.44
CA9 Q16790 1/20 0.44
PARP1 P09874 3/20 0.42
PDPK1 O15530 1/20 0.42
PARP10 Q53GL7 1/20 0.42
PARP11 Q9NR21 1/20 0.42
TDP2 O95551 1/20 0.42
CASP3 P42574 1/20 0.42
CASP7 P55210 1/20 0.42
CASP9 P55211 1/20 0.42
CASP6 P55212 1/20 0.42
CASP8 Q14790 1/20 0.42
MAP3K14 Q99558 1/20 0.42
ACHE P22303 1/20 0.42
MAOA P21397 1/20 0.39
CYP19A1 P11511 2/20 0.38
DYRK1A Q13627 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TNKS2 Q9H2K2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446225 0.84 TSHR (0.57) TSHRCA12CA9PARP1PDPK1
SCHEMBL7439402 0.83 TSHR (0.47) TSHRCA12CA9PARP1PDPK1
SCHEMBL22799646 0.80 TSHR (0.40) TSHRCA12CA9PARP1PDPK1
SCHEMBL22799721 0.78 CYP2A6 (0.45) TSHRCA12CA9PARP1PDPK1
SCHEMBL22799901 0.78 CYP2A6 (0.45) TSHRCA12CA9PARP1PDPK1
SCHEMBL22799843 0.78 CYP2A6 (0.45) TSHRCA12CA9PARP1PDPK1
SCHEMBL348705 0.76 MAPT (0.50) TSHR
SCHEMBL7551415 0.76 MAPT (0.50) TSHR
SCHEMBL14306724 0.76 MAPT (0.50) TSHR
SCHEMBL7444393 0.75 ANPEP (0.41) TSHRPARP1TDP2CASP3CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098888-A Cholinergic agents and antispasmodic agents ADIR ET COMPAGNIE (FR) 1992-03-24 US disclosed