SCHEMBL9733426

SCHEMBL9733426

COC(=O)C(C)(C)CC(=O)c1ccc(OC)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.66
ALDH1A1 P00352 3/20 0.61
LMNA P02545 1/20 0.61
ALOX15 P16050 1/20 0.61
APEX1 P27695 1/20 0.61
MAPK1 P28482 1/20 0.61
RECQL P46063 1/20 0.61
HSD17B10 Q99714 1/20 0.61
TDP1 Q9NUW8 1/20 0.61
HDAC1 Q13547 4/20 0.56
HDAC8 Q9BY41 4/20 0.56
HDAC3 O15379 2/20 0.56
HDAC4 P56524 2/20 0.56
HDAC7 Q8WUI4 2/20 0.56
HDAC2 Q92769 2/20 0.56
HDAC10 Q969S8 2/20 0.56
HDAC11 Q96DB2 2/20 0.56
HDAC6 Q9UBN7 2/20 0.56
HDAC9 Q9UKV0 2/20 0.56
HDAC5 Q9UQL6 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7902328 0.84 ALDH1A1 (0.62) GAAALDH1A1LMNAALOX15APEX1
SCHEMBL1748024 0.83 GSK3B (0.48) GAAALDH1A1LMNAALOX15APEX1
SCHEMBL12121918 0.83 GSK3B (0.48) GAAALDH1A1LMNAMAPK1GSK3B
SCHEMBL380738 0.82 SRC (0.53) GAAALDH1A1LMNAALOX15MAPK1
SCHEMBL4095875 0.80 ALDH1A1 (0.54) GAAALDH1A1LMNAALOX15APEX1
SCHEMBL153386 0.79 ALDH1A1 (0.76) ALDH1A1LMNAALOX15APEX1MAPK1
SCHEMBL595610 0.79 GAA (0.43) GAAALDH1A1LMNAALOX15APEX1
SCHEMBL29434793 0.79 GAA (0.65) GAAALDH1A1LMNAALOX15APEX1
SCHEMBL821204 0.78 GAA (0.47) GAAALDH1A1LMNAALOX15APEX1
Hydrochloric Acid SCHEMBL7011412 0.78 ALDH1A1 (0.55) GAAALDH1A1LMNAALOX15APEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135940-A Antiallegens, antiinflammatory agents MERCK FROSST CANADA, INC. (CA) 1992-08-04 US disclosed
EP-0252639-A1 Leukotriene antagonists MERCK FROSST CANADA INC. (CA) 1988-01-13 EP disclosed
EP-0104885-B1 LEUKOTRIENE ANTAGONISTS, THEIR PRODUCTION, AND COMPOSITIONS CONTAINING THEM MERCK FROSST CANADA INC. (CA) 1986-06-04 EP disclosed
EP-0104885-A1 Leukotriene antagonists, their production, and compositions containing them MERCK FROSST CANADA INC. (CA) 1984-04-04 EP disclosed