SCHEMBL9733990

SCHEMBL9733990

COc1cccc2c1CC(NC(=O)c1ccccc1)CC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 8/20 1.00
MTNR1B P49286 8/20 1.00
CYP1A2 P05177 1/20 0.68
MAPT P10636 1/20 0.68
CYP2C9 P11712 1/20 0.68
ALOX15 P16050 1/20 0.68
CA1 P00915 2/20 0.58
CA2 P00918 2/20 0.58
ACHE P22303 2/20 0.58
EPHX2 P34913 1/20 0.54
ADORA2A P29274 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6518723 0.90 MTNR1A (0.82) MTNR1AMTNR1BCYP1A2MAPTCYP2C9
SCHEMBL6518717 0.90 MTNR1A (0.82) MTNR1AMTNR1BCYP1A2MAPTCYP2C9
SCHEMBL3919777 0.84 MTNR1A (1.00) MTNR1AMTNR1BCYP1A2MAPTCYP2C9
SCHEMBL10447045 0.83 MTNR1A (0.70) MTNR1AMTNR1B
SCHEMBL55491 0.82 MTNR1A (1.00) MTNR1AMTNR1BCYP1A2MAPTCYP2C9
SCHEMBL81120 0.82 MTNR1A (1.00) MTNR1AMTNR1BCYP1A2MAPTCYP2C9
SCHEMBL6516803 0.82 MTNR1A (0.70) MTNR1AMTNR1BCYP1A2MAPTCYP2C9
SCHEMBL6513612 0.82 MTNR1A (0.70) MTNR1AMTNR1BCYP1A2MAPTCYP2C9
SCHEMBL6513609 0.82 MTNR1A (0.70) MTNR1AMTNR1BCYP1A2MAPTCYP2C9
Hydrochloric Acid SCHEMBL27339226 0.81 MTNR1A (0.68) MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5151446-A Neurological disorders or cardiovascular disorders NORTHWESTERN UNIVERSITY (US) 1992-09-29 US disclosed
US-5071875-A Nervous system, psychological disorders; sleep cycle, skin dis coloration NORTHWESTERN UNIVERSITY (US) 1991-12-10 US disclosed
EP-0420064-A2 Substituted 2-amidotetralins as melatonin agonists and antagonists NORTHWESTERN UNIVERSITY (US) 1991-04-03 EP disclosed