SCHEMBL9734283

SCHEMBL9734283

CCOC(=O)CC(C#N)(C(=O)OCC)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.47
PIN1 Q13526 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
POLB P06746 3/20 0.42
HSD11B1 P28845 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TSHR P16473 1/20 0.40
PPID Q08752 1/20 0.40
ALDH1A1 P00352 3/20 0.39
RECQL P46063 1/20 0.39
MMP8 P22894 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
NLRP3 Q96P20 1/20 0.39
KCNA3 P22001 1/20 0.38
OPRM1 P35372 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9214363 0.87 CCR1 (0.50) CCR1PIN1SMN1; SMN2POLBNPSR1
SCHEMBL2516644 0.86 MAPT (0.41) CCR1SMN1; SMN2POLBNPSR1ALDH1A1
SCHEMBL1625711 0.85 CCR1 (0.48) CCR1PIN1POLBTDP1NPSR1
SCHEMBL27450756 0.84 CCR1 (0.48) CCR1PIN1SMN1; SMN2POLBNPSR1
SCHEMBL9734250 0.84 CCR1 (0.54) CCR1PIN1SMN1; SMN2POLBALDH1A1
SCHEMBL8311559 0.82 OPRM1 (0.49) SMN1; SMN2POLBHSD11B1TDP1TSHR
SCHEMBL22323105 0.82 CCR1 (0.54) CCR1PIN1SMN1; SMN2POLBNPSR1
SCHEMBL2636117 0.81 SMN1; SMN2 (0.46) SMN1; SMN2POLBHSD11B1TDP1PPID
SCHEMBL22323061 0.81 CCR1 (0.46) CCR1PIN1SMN1; SMN2POLBNPSR1
SCHEMBL18153522 0.80 SMN1; SMN2 (0.48) CCR1SMN1; SMN2POLBNPSR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5164386-A Gastrointestinal and respiratory disorders ISTITUTO DE ANGELI S.P.A. (IT) 1992-11-17 US disclosed
EP-0404737-A2 New R(-) 3-quinuclidinol derivatives BOEHRINGER INGELHEIM ITALIA S.p.A. (IT) 1990-12-27 EP disclosed