SCHEMBL9734614

SCHEMBL9734614

CC(C(=O)O)c1ccc2c(c1)OCc1ccccc1C2=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.58
MAPK14 Q16539 7/20 0.52
PTGS1 P23219 1/20 0.51
PTGS2 P35354 1/20 0.51
SMN1; SMN2 Q16637 3/20 0.49
TP53 P04637 2/20 0.49
RAB9A P51151 2/20 0.49
ALDH1A1 P00352 2/20 0.49
MAPT P10636 2/20 0.49
MEN1 O00255 1/20 0.49
LMNA P02545 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C19 P33261 1/20 0.49
KMT2A Q03164 1/20 0.49
NPC1 O15118 1/20 0.49
PGR P06401 1/20 0.49
CYP3A4 P08684 1/20 0.49
GAA P10253 1/20 0.49
PKM P14618 1/20 0.49
NFKB1 P19838 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9222163 0.90 MAPT (0.59) PTGS1PTGS2SMN1; SMN2RAB9AALDH1A1
SCHEMBL11179898 0.85 AKR1B1 (0.54) AKR1B1MAPK14SMN1; SMN2RAB9AALDH1A1
Water SCHEMBL10842921 0.83 MAPT (0.52) SMN1; SMN2RAB9AALDH1A1MAPTKMT2A
SCHEMBL11834532 0.81 AKR1B1 (0.68) AKR1B1MAPK14PTGS1PTGS2SMN1; SMN2
SCHEMBL12726875 0.79 AKR1C3 (0.59) AKR1B1PTGS1PTGS2SMN1; SMN2ALDH1A1
SCHEMBL12726876 0.79 AKR1B1 (0.54) AKR1B1PTGS1PTGS2SMN1; SMN2TP53
SCHEMBL9210700 0.79 ALDH1A1 (0.58) SMN1; SMN2RAB9AALDH1A1MAPTKMT2A
SCHEMBL15195012 0.78 PTGS1 (0.51) AKR1B1PTGS1PTGS2ALDH1A1MAPT
SCHEMBL11189383 0.78 MAPT (0.60) AKR1B1MAPK14SMN1; SMN2RAB9AALDH1A1
SCHEMBL12726878 0.77 AKR1C3 (0.58) AKR1B1PTGS1PTGS2SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-55000377-A None JP disclosed
US-5175286-A Antiphlogistic agent HISAMITSU PHARMACEUTICAL CO., INC. (JP) 1992-12-29 US disclosed
EP-0436025-A1 NOVEL DIBENZ b,e]OXEPIN DERIVATIVES Hisamitsu Pharmaceutical Co., Inc. (JP) 1991-07-10 EP disclosed
US-4292319-A MIXTURE WITH AN ANTIULCER AGENT BOEHRINGER INGELHEIM GMBH (DE) 1981-09-29 US disclosed
US-4256747-A ANTIINFLAMMATORY AGENTS, PYRIDO/2,3B//1,4/BENZODIAZEPIN-6-ONES BOEHRINGER INGELHEIM GMBH (DE) 1981-03-17 US disclosed
JP-S55377-A PREPARATION OF DIBENZOXEPIN DERIVATIVE DAI ICHI SEIYAKU CO LTD 1980-01-05 JP disclosed
US-4154833-A INDOMETHACIN (1-(4-CHLOROBENZOYL)-5-METHOXY-2-METHYL-1H-INDOLE-3-ACETIC ACID) WITH PIRENZEPINE (5,11-DIHYDRO-11-((4-METHYL-1-PIPERAZINYL)-ACETYL)-6H-PYRIDO(2,3 -B)(1,4)BENZODIAZEPIN-6-ONE) BOEHRINGER INGELHEIM GMBH (DE) 1979-05-15 US disclosed