SCHEMBL9734722

SCHEMBL9734722

O=C(C1CC2(CCN1)OCCO2)N1CCCC1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.43
CYP2C19 P33261 2/20 0.38
ALDH1A1 P00352 5/20 0.37
DPP4 P27487 2/20 0.35
HRH3 Q9Y5N1 5/20 0.35
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 2/20 0.35
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
DPP8 Q6V1X1 1/20 0.34
DPP9 Q86TI2 1/20 0.34
HDAC2 Q92769 1/20 0.34
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733467 0.82 NPC1 (0.33) CYP2C19ALDH1A1
SCHEMBL27172650 0.77 CYP1A2 (0.38) CYP2C19ALDH1A1LMNAKMT2ATSHR
SCHEMBL16894869 0.77 CYP1A2 (0.38) CYP2C19ALDH1A1LMNAKMT2ATSHR
SCHEMBL15152229 0.77 CYP1A2 (0.38) CYP2C19ALDH1A1LMNAKMT2ATSHR
SCHEMBL9192107 0.76 DPP4 (0.41) HPGDDPP4HRH3KMT2AL3MBTL1
SCHEMBL9733517 0.72 MMP2 (0.35) KMT2A
SCHEMBL10466402 0.69 DPP4 (0.40) HPGDALDH1A1DPP4KMT2ADPP8
SCHEMBL488954 0.68 DPP4 (0.64) HPGDDPP4L3MBTL1DPP8DPP9
SCHEMBL1383434 0.68 DPP4 (0.64) HPGDDPP4L3MBTL1DPP8DPP9
SCHEMBL488953 0.68 DPP4 (0.64) HPGDDPP4L3MBTL1DPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5114945-A Spiropiperidine derivatives GLAXO GROUP LIMITED (GB) 1992-05-19 US disclosed
EP-0330461-A2 Piperidine derivatives GLAXO GROUP LIMITED (GB) 1989-08-30 EP disclosed